Detalhe da pesquisa
1.
Design, evaluation, and comparison of ghrelin receptor agonists and inverse agonists as suitable radiotracers for PET imaging.
Bioconjug Chem
; 23(4): 771-84, 2012 Apr 18.
Artigo
Inglês
| MEDLINE | ID: mdl-22372770
2.
Development of a ghrelin receptor inverse agonist for positron emission tomography.
Oncotarget
; 12(5): 450-474, 2021 Mar 02.
Artigo
Inglês
| MEDLINE | ID: mdl-33747360
3.
Targeted delivery of compounds to Trypanosoma brucei using the melamine motif.
Bioorg Med Chem
; 17(6): 2512-23, 2009 Mar 15.
Artigo
Inglês
| MEDLINE | ID: mdl-19250832
4.
Ghrelin--a novel generation of anti-obesity drug: design, pharmacomodulation and biological activity of ghrelin analogues.
J Pept Sci
; 15(11): 711-30, 2009 Nov.
Artigo
Inglês
| MEDLINE | ID: mdl-19787814
5.
In vitro antileishmanial activity of fluoro-artemisinin derivatives against Leishmania donovani.
Biomed Pharmacother
; 62(7): 462-5, 2008 Sep.
Artigo
Inglês
| MEDLINE | ID: mdl-18538529
6.
Development of Substrate-Derived Sirtuin Inhibitors with Potential Anticancer Activity.
ChemMedChem
; 12(20): 1703-1714, 2017 10 20.
Artigo
Inglês
| MEDLINE | ID: mdl-28776959
7.
Rational design of dual peptides targeting ghrelin and Y2 receptors to regulate food intake and body weight.
J Med Chem
; 58(10): 4180-93, 2015 May 28.
Artigo
Inglês
| MEDLINE | ID: mdl-25905598
8.
Integrating solid-state NMR and computational modeling to investigate the structure and dynamics of membrane-associated ghrelin.
PLoS One
; 10(3): e0122444, 2015.
Artigo
Inglês
| MEDLINE | ID: mdl-25803439
9.
An aromatic region to induce a switch between agonism and inverse agonism at the ghrelin receptor.
J Med Chem
; 55(17): 7437-49, 2012 Sep 13.
Artigo
Inglês
| MEDLINE | ID: mdl-22920150
10.
Ghrelin receptor: high constitutive activity and methods for developing inverse agonists.
Methods Enzymol
; 485: 103-21, 2010.
Artigo
Inglês
| MEDLINE | ID: mdl-21050913
11.
S(N)/S(N)' competition: selective access to new 10-fluoro artemisinins.
J Org Chem
; 71(8): 3082-5, 2006 Apr 14.
Artigo
Inglês
| MEDLINE | ID: mdl-16599603