Detalhe da pesquisa
1.
Optimization of M4 positive allosteric modulators (PAMs): The discovery of VU0476406, a non-human primate in vivo tool compound for translational pharmacology.
Bioorg Med Chem Lett
; 27(11): 2296-2301, 2017 06 01.
Artigo
Inglês
| MEDLINE | ID: mdl-28442253
2.
Discovery of VU6005649, a CNS Penetrant mGlu7/8 Receptor PAM Derived from a Series of Pyrazolo[1,5-a]pyrimidines.
ACS Med Chem Lett
; 8(10): 1110-1115, 2017 Oct 12.
Artigo
Inglês
| MEDLINE | ID: mdl-29057060
3.
VU6010608, a Novel mGlu7 NAM from a Series of N-(2-(1H-1,2,4-Triazol-1-yl)-5-(trifluoromethoxy)phenyl)benzamides.
ACS Med Chem Lett
; 8(12): 1326-1330, 2017 Dec 14.
Artigo
Inglês
| MEDLINE | ID: mdl-29259756