Detalhe da pesquisa
1.
Impact of dipeptide on ADC physicochemical properties and efficacy identifies Ala-Ala as the optimal dipeptide.
RSC Med Chem
; 15(1): 355-365, 2024 Jan 25.
Artigo
Inglês
| MEDLINE | ID: mdl-38283215
2.
Linker substitution influences succinimide ring hydrolysis equilibrium impacting the stability of attachment to antibody-drug conjugates.
RSC Med Chem
; 15(2): 612-622, 2024 Feb 21.
Artigo
Inglês
| MEDLINE | ID: mdl-38389885
3.
Anti-TNF Thioester Glucocorticoid Antibody-Drug Conjugate Fully Inhibits Inflammation with Minimal Effect on Systemic Corticosterone Levels in a Mouse Arthritis Model.
J Med Chem
; 67(11): 9495-9515, 2024 Jun 13.
Artigo
Inglês
| MEDLINE | ID: mdl-38780432
4.
Optimization of Drug-Linker to Enable Long-term Storage of Antibody-Drug Conjugate for Subcutaneous Dosing.
J Med Chem
; 66(13): 9161-9173, 2023 07 13.
Artigo
Inglês
| MEDLINE | ID: mdl-37379257
5.
Discovery of ABBV-154, an anti-TNF Glucocorticoid Receptor Modulator Immunology Antibody-Drug Conjugate (iADC).
J Med Chem
; 66(17): 12544-12558, 2023 09 14.
Artigo
Inglês
| MEDLINE | ID: mdl-37656698
6.
Design and Development of Glucocorticoid Receptor Modulators as Immunology Antibody-Drug Conjugate Payloads.
J Med Chem
; 65(6): 4500-4533, 2022 03 24.
Artigo
Inglês
| MEDLINE | ID: mdl-35133822
7.
Discovery of ABBV-3373, an Anti-TNF Glucocorticoid Receptor Modulator Immunology Antibody Drug Conjugate.
J Med Chem
; 65(23): 15893-15934, 2022 12 08.
Artigo
Inglês
| MEDLINE | ID: mdl-36394224
8.
Novel approach to optimization of a high-throughput semipreparative LC/MS system.
J Comb Chem
; 11(4): 592-7, 2009.
Artigo
Inglês
| MEDLINE | ID: mdl-19422189
9.
Correction to "Design and Development of Glucocorticoid Receptor Modulators as Immunology Antibody-Drug Conjugate Payloads".
J Med Chem
; 66(8): 6011, 2023 Apr 27.
Artigo
Inglês
| MEDLINE | ID: mdl-37058612
10.
Correction to "Discovery of ABBV-3373, an Anti-TNF Glucocorticoid Receptor Modulator Immunology Antibody Drug Conjugate".
J Med Chem
; 66(8): 6010, 2023 Apr 27.
Artigo
Inglês
| MEDLINE | ID: mdl-37027784