Detalhe da pesquisa
1.
Genotoxicity assessment of four novel quinazoline-derived trypanocidal agents in the Drosophila wing somatic mutation and recombination test.
Mutagenesis
; 35(4): 299-310, 2020 09 12.
Artigo
Inglês
| MEDLINE | ID: mdl-31793639
2.
Evaluation of New Benzimidazole Derivatives as Cysticidal Agents: In Vitro, in Vivo and Docking Studies.
Chem Pharm Bull (Tokyo)
; 67(12): 1293-1300, 2019.
Artigo
Inglês
| MEDLINE | ID: mdl-31787656
3.
Systematic search for benzimidazole compounds and derivatives with antileishmanial effects.
Mol Divers
; 22(4): 779-790, 2018 Nov.
Artigo
Inglês
| MEDLINE | ID: mdl-29748853
4.
Synthesis and biological evaluation of 2-methyl-1H-benzimidazole-5-carbohydrazides derivatives as modifiers of redox homeostasis of Trypanosoma cruzi.
Bioorg Med Chem Lett
; 27(15): 3403-3407, 2017 08 01.
Artigo
Inglês
| MEDLINE | ID: mdl-28648464
5.
Species-Specific Inactivation of Triosephosphate Isomerase from Trypanosoma brucei: Kinetic and Molecular Dynamics Studies.
Molecules
; 22(12)2017 11 24.
Artigo
Inglês
| MEDLINE | ID: mdl-29186784
6.
Synthesis and molecular docking of N'-arylidene-5-(4-chlorophenyl)-1-(3,4-dichlorophenyl)-4-methyl-1H-pyrazole-3-carbohydrazides as novel hypoglycemic and antioxidant dual agents.
Bioorg Med Chem
; 24(10): 2298-306, 2016 05 15.
Artigo
Inglês
| MEDLINE | ID: mdl-27079123
7.
JVG9, a benzimidazole derivative, alters the surface and cytoskeleton of Trypanosoma cruzi bloodstream trypomastigotes.
Mem Inst Oswaldo Cruz
; 109(6): 757-60, 2014 Sep.
Artigo
Inglês
| MEDLINE | ID: mdl-25317703
8.
Compounds Consisting of Quinazoline, Ibuprofen, and Amino Acids with Cytotoxic and Anti-Inflammatory Effects.
ChemMedChem
; 19(10): e202300651, 2024 May 17.
Artigo
Inglês
| MEDLINE | ID: mdl-38354370
9.
Effects of an antimalarial quinazoline derivative on human erythrocytes and on cell membrane molecular models.
Biochim Biophys Acta
; 1818(3): 738-46, 2012 Mar.
Artigo
Inglês
| MEDLINE | ID: mdl-22155684
10.
Synthesis and antiprotozoal activity of novel 2-{[2-(1H-imidazol-1-yl)ethyl]sulfanyl}-1H-benzimidazole derivatives.
Bioorg Med Chem Lett
; 23(14): 4221-4, 2013 Jul 15.
Artigo
Inglês
| MEDLINE | ID: mdl-23731944
11.
Synthesis and antiprotozoal activity of nitazoxanide-N-methylbenzimidazole hybrids.
Bioorg Med Chem Lett
; 23(24): 6838-41, 2013 Dec 15.
Artigo
Inglês
| MEDLINE | ID: mdl-24183540
12.
RCB20, an experimental benzimidazole derivative, affects tubulin expression and induces gross anatomical changes in Taenia crassiceps cysticerci.
Parasitol Res
; 112(6): 2215-26, 2013 Jun.
Artigo
Inglês
| MEDLINE | ID: mdl-23504054
13.
Albendazole and its derivative JVG9 induce encystation on Giardia intestinalis trophozoites.
Parasitol Res
; 112(9): 3251-7, 2013 Sep.
Artigo
Inglês
| MEDLINE | ID: mdl-23857298
14.
Synthesis of Quinazolin-2,4,6-triamine Derivatives as Non-purine Xanthine Oxidase Inhibitors and Exploration of Their Toxicological Potential.
ChemMedChem
; 18(20): e202300184, 2023 10 17.
Artigo
Inglês
| MEDLINE | ID: mdl-37642254
15.
Antiprotozoal activity of proton-pump inhibitors.
Bioorg Med Chem Lett
; 21(24): 7351-4, 2011 Dec 15.
Artigo
Inglês
| MEDLINE | ID: mdl-22047694
16.
Studies on 6-chloro-5-(1-naphthyloxy)-2-(trifluoromethyl)-1H-benzimidazole/2-hydroxypropyl-ß-cyclodextrin association: Characterization, molecular modeling studies, and in vivo anthelminthic activity.
Bioorg Med Chem
; 19(2): 789-97, 2011 Jan 15.
Artigo
Inglês
| MEDLINE | ID: mdl-21190860
17.
In Silico Characterization of Masitinib Interaction with SARS-CoV-2 Main Protease.
ChemMedChem
; 16(15): 2339-2344, 2021 08 05.
Artigo
Inglês
| MEDLINE | ID: mdl-34142459
18.
Design, Synthesis and Evaluation of 2,4-Diaminoquinazoline Derivatives as Potential Tubulin Polymerization Inhibitors.
ChemMedChem
; 15(19): 1802-1812, 2020 10 05.
Artigo
Inglês
| MEDLINE | ID: mdl-32686342
19.
Synthesis and antiprotozoal activity of novel 1-methylbenzimidazole derivatives.
Bioorg Med Chem
; 17(4): 1724-30, 2009 Feb 15.
Artigo
Inglês
| MEDLINE | ID: mdl-19186059
20.
Synthesis and antiprotozoal activity of some 2-(trifluoromethyl)-1H-benzimidazole bioisosteres.
Eur J Med Chem
; 41(1): 135-41, 2006 Jan.
Artigo
Inglês
| MEDLINE | ID: mdl-16260067