Detalhe da pesquisa
1.
Cholesteryl ester transfer protein (CETP) inhibitors based on cyclic urea, bicyclic urea and bicyclic sulfamide cores.
Bioorg Med Chem Lett
; 32: 127668, 2021 01 15.
Artigo
Inglês
| MEDLINE | ID: mdl-33161125
2.
Potent, non-covalent reversible BTK inhibitors with 8-amino-imidazo[1,5-a]pyrazine core featuring 3-position bicyclic ring substitutes.
Bioorg Med Chem Lett
; 30(17): 127390, 2020 09 01.
Artigo
Inglês
| MEDLINE | ID: mdl-32738973
3.
Accelerating the discovery of DGAT1 inhibitors through the application of parallel medicinal chemistry (PMC).
Bioorg Med Chem Lett
; 29(11): 1380-1385, 2019 06 01.
Artigo
Inglês
| MEDLINE | ID: mdl-30952592
4.
Benzimidazole-based DGAT1 inhibitors with a [3.1.0] bicyclohexane carboxylic acid moiety.
Bioorg Med Chem Lett
; 29(10): 1182-1186, 2019 05 15.
Artigo
Inglês
| MEDLINE | ID: mdl-30926247
5.
Discovery of novel BTK inhibitors with carboxylic acids.
Bioorg Med Chem Lett
; 27(6): 1471-1477, 2017 03 15.
Artigo
Inglês
| MEDLINE | ID: mdl-28254166
6.
Discovery of 3-morpholino-imidazole[1,5-a]pyrazine BTK inhibitors for rheumatoid arthritis.
Bioorg Med Chem Lett
; 27(16): 3939-3943, 2017 08 15.
Artigo
Inglês
| MEDLINE | ID: mdl-28720503
7.
Discovery of 8-Amino-imidazo[1,5-a]pyrazines as Reversible BTK Inhibitors for the Treatment of Rheumatoid Arthritis.
ACS Med Chem Lett
; 7(2): 198-203, 2016 Feb 11.
Artigo
Inglês
| MEDLINE | ID: mdl-26985298
8.
Discovery of a Potent and Selective DGAT1 Inhibitor with a Piperidinyl-oxy-cyclohexanecarboxylic Acid Moiety.
ACS Med Chem Lett
; 5(10): 1082-7, 2014 Oct 09.
Artigo
Inglês
| MEDLINE | ID: mdl-25349648
9.
Potent DGAT1 Inhibitors in the Benzimidazole Class with a Pyridyl-oxy-cyclohexanecarboxylic Acid Moiety.
ACS Med Chem Lett
; 4(8): 773-8, 2013 Aug 08.
Artigo
Inglês
| MEDLINE | ID: mdl-24900745