Detalhe da pesquisa
1.
Synthesis of new compounds bearing methyl sulfonyl pharmacophore as selective COX-2 inhibitor.
J Mol Recognit
; 36(7): e3025, 2023 07.
Artigo
Inglês
| MEDLINE | ID: mdl-37191245
2.
Design, synthesis, biological activities, and evaluation of molecular docking-dynamics studies of new thiosemicarbazones that may be effective against Alzheimer's disease.
J Mol Recognit
; 36(12): e3059, 2023 12.
Artigo
Inglês
| MEDLINE | ID: mdl-37723924
3.
Synthesis of Imidazole-2,3-dihydrothiazole Compounds as VEGFR-2 Inhibitors and Their Support with in Silico Studies.
Chem Biodivers
; 20(9): e202300944, 2023 Sep.
Artigo
Inglês
| MEDLINE | ID: mdl-37503680
4.
Synthesis of novel thiosemicarbazone derivatives and investigation of their dual AChE and MAO-B inhibitor effects.
J Mol Recognit
; 35(12): e2990, 2022 12.
Artigo
Inglês
| MEDLINE | ID: mdl-36056718
5.
Design, synthesis, molecular docking and molecular dynamics studies of novel triazolothiadiazine derivatives containing furan or thiophene rings as anticancer agents.
Bioorg Chem
; 122: 105709, 2022 05.
Artigo
Inglês
| MEDLINE | ID: mdl-35255344
6.
Synthesis of New Pyrimidine-Triazole Derivatives and Investigation of Their Anticancer Activities.
Chem Biodivers
; 19(8): e202200216, 2022 Aug.
Artigo
Inglês
| MEDLINE | ID: mdl-35699405
7.
Design, synthesis, and biological activity of novel dithiocarbamate-methylsulfonyl hybrids as carbonic anhydrase inhibitors.
Arch Pharm (Weinheim)
; 355(8): e2200132, 2022 Aug.
Artigo
Inglês
| MEDLINE | ID: mdl-35502846
8.
Design and synthesis of novel chalcone derivatives and evaluation of their inhibitory activities against acetylcholinesterase.
Arch Pharm (Weinheim)
; 355(3): e2100372, 2022 Mar.
Artigo
Inglês
| MEDLINE | ID: mdl-34893996
9.
Design, synthesis, biological activity, molecular docking, and molecular dynamics of novel benzimidazole derivatives as potential AChE/MAO-B dual inhibitors.
Arch Pharm (Weinheim)
; 355(3): e2100450, 2022 Mar.
Artigo
Inglês
| MEDLINE | ID: mdl-34931332
10.
Design, Synthesis, and Evaluation of Novel 2H-Benzo[b][1,4]thiazin-3(4H)-one Derivatives as New Acetylcholinesterase Inhibitors.
Molecules
; 27(7)2022 Mar 25.
Artigo
Inglês
| MEDLINE | ID: mdl-35408519
11.
Design, synthesis, in vitro, and in silico studies of 1,2,4-triazole-piperazine hybrid derivatives as potential MAO inhibitors.
Bioorg Chem
; 117: 105430, 2021 12.
Artigo
Inglês
| MEDLINE | ID: mdl-34678603
12.
Design, synthesis, in vitro and in silico studies of some novel thiazole-dihydrofuran derivatives as aromatase inhibitors.
Bioorg Chem
; 114: 105123, 2021 09.
Artigo
Inglês
| MEDLINE | ID: mdl-34214753
13.
Design, Synthesis and Biological Evaluation of New N-Acyl Hydrazones with a Methyl Sulfonyl Moiety as Selective COX-2 Inhibitors.
Chem Biodivers
; 18(11): e2100521, 2021 Nov.
Artigo
Inglês
| MEDLINE | ID: mdl-34411436
14.
Design, synthesis, biological evaluation, and docking studies of some novel chalcones as selective COX-2 inhibitors.
Arch Pharm (Weinheim)
; 354(3): e2000273, 2021 Mar.
Artigo
Inglês
| MEDLINE | ID: mdl-33244799
15.
Novel Thiosemicarbazone Derivatives: In Vitro and In Silico Evaluation as Potential MAO-B Inhibitors.
Molecules
; 26(21)2021 Nov 02.
Artigo
Inglês
| MEDLINE | ID: mdl-34771054
16.
Synthesis and Antinociceptive Effect of Some Thiazole-Piperazine Derivatives: Involvement of Opioidergic System in the Activity.
Molecules
; 26(11)2021 Jun 02.
Artigo
Inglês
| MEDLINE | ID: mdl-34199486
17.
Synthesis, anticancer evaluation and molecular docking studies of new benzimidazole- 1,3,4-oxadiazole derivatives as human topoisomerase types I poison.
J Enzyme Inhib Med Chem
; 35(1): 1657-1673, 2020 Dec.
Artigo
Inglês
| MEDLINE | ID: mdl-32811204
18.
Synthesis, in vitro enzyme activity and molecular docking studies of new benzylamine-sulfonamide derivatives as selective MAO-B inhibitors.
J Enzyme Inhib Med Chem
; 35(1): 1422-1432, 2020 Dec.
Artigo
Inglês
| MEDLINE | ID: mdl-32602377
19.
Synthesis and docking study of benzimidazole-triazolothiadiazine hybrids as aromatase inhibitors.
Arch Pharm (Weinheim)
; 353(5): e2000008, 2020 May.
Artigo
Inglês
| MEDLINE | ID: mdl-32159244
20.
Design, Synthesis, and Structure-Activity Relationships of Thiazole Analogs as Anticholinesterase Agents for Alzheimer's Disease.
Molecules
; 25(18)2020 Sep 20.
Artigo
Inglês
| MEDLINE | ID: mdl-32962239