Detalhe da pesquisa
1.
Knock-in mutagenesis in Drosophila Rdl underscores the critical role of the conserved M3 glycine in mediating the actions of broflanilide and isocycloseram on GABA receptors.
Pestic Biochem Physiol
; 199: 105776, 2024 Feb.
Artigo
Inglês
| MEDLINE | ID: mdl-38458683
2.
Controlled expression of nicotinic acetylcholine receptor-encoding genes in insects uncovers distinct mechanisms of action of the neonicotinoid insecticide dinotefuran.
Pestic Biochem Physiol
; 191: 105378, 2023 Apr.
Artigo
Inglês
| MEDLINE | ID: mdl-36963946
3.
State-dependent inhibition of GABA receptor channels by the ectoparasiticide fluralaner.
Pestic Biochem Physiol
; 181: 105008, 2022 Feb.
Artigo
Inglês
| MEDLINE | ID: mdl-35082031
4.
Ion channels and G protein-coupled receptors as targets for invertebrate pest control: from past challenges to practical insecticides.
Biosci Biotechnol Biochem
; 85(7): 1563-1571, 2021 Jun 24.
Artigo
Inglês
| MEDLINE | ID: mdl-33988673
5.
Structure-dependent receptor subtype selectivity and G protein subtype preference of heterocyclic agonists in heterologously expressed silkworm octopamine receptors.
Pestic Biochem Physiol
; 177: 104895, 2021 Aug.
Artigo
Inglês
| MEDLINE | ID: mdl-34301357
6.
Further characterization of distinct high-affinity binding sites for dinotefuran in the abdominal nerve cord of the American cockroach Periplaneta americana (Blattodea).
Pestic Biochem Physiol
; 165: 104554, 2020 May.
Artigo
Inglês
| MEDLINE | ID: mdl-32359545
7.
Effects of intersubunit amino acid substitutions on GABA receptor sensitivity to the ectoparasiticide fluralaner.
Pestic Biochem Physiol
; 163: 123-129, 2020 Feb.
Artigo
Inglês
| MEDLINE | ID: mdl-31973848
8.
4-Aryl-5-carbamoyl-3-isoxazolols as competitive antagonists of insect GABA receptors: Synthesis, biological activity, and molecular docking studies.
Bioorg Med Chem
; 27(2): 416-424, 2019 01 15.
Artigo
Inglês
| MEDLINE | ID: mdl-30579800
9.
Spatiotemporally different expression of alternatively spliced GABA receptor subunit transcripts in the housefly Musca domestica.
Arch Insect Biochem Physiol
; 101(1): e21541, 2019 May.
Artigo
Inglês
| MEDLINE | ID: mdl-30821008
10.
Fluxametamide: A novel isoxazoline insecticide that acts via distinctive antagonism of insect ligand-gated chloride channels.
Pestic Biochem Physiol
; 151: 67-72, 2018 Oct.
Artigo
Inglês
| MEDLINE | ID: mdl-30704715
11.
A Single Amino Acid Substitution in the Third Transmembrane Region Has Opposite Impacts on the Selectivity of the Parasiticides Fluralaner and Ivermectin for Ligand-Gated Chloride Channels.
Mol Pharmacol
; 92(5): 546-555, 2017 11.
Artigo
Inglês
| MEDLINE | ID: mdl-28887352
12.
Synthesis of photoreactive ivermectin B1a derivatives and their actions on Haemonchus and Bombyx glutamate-gated chloride channels.
Pestic Biochem Physiol
; 120: 82-90, 2015 May.
Artigo
Inglês
| MEDLINE | ID: mdl-25987225
13.
Competitive antagonism of insect GABA receptors by 4-substituted 5-(4-piperidyl)-3-isothiazolols.
Bioorg Med Chem
; 22(17): 4637-45, 2014 Sep 01.
Artigo
Inglês
| MEDLINE | ID: mdl-25112550
14.
Mechanistic insights into the selectivity of bicyclophosphorothionate antagonists for housefly versus rat GABA receptors.
Pest Manag Sci
; 80(3): 1382-1399, 2024 Mar.
Artigo
Inglês
| MEDLINE | ID: mdl-37926485
15.
Electrophysiological evidence for 4-isobutyl-3-isopropylbicyclophosphorothionate as a selective blocker of insect GABA-gated chloride channels.
Bioorg Med Chem Lett
; 23(11): 3373-6, 2013 Jun 01.
Artigo
Inglês
| MEDLINE | ID: mdl-23591113
16.
Insecticidal 3-benzamido-N-phenylbenzamides specifically bind with high affinity to a novel allosteric site in housefly GABA receptors.
Pestic Biochem Physiol
; 107(3): 285-92, 2013 Nov.
Artigo
Inglês
| MEDLINE | ID: mdl-24267689
17.
External amino acid residues of insect GABA receptor channels dictate the action of the isoxazoline ectoparasiticide fluralaner.
Pest Manag Sci
; 79(10): 4078-4082, 2023 Oct.
Artigo
Inglês
| MEDLINE | ID: mdl-37288963
18.
A glutamate-gated chloride channel as the mite-specific target-site of dicofol and other diphenylcarbinol acaricides.
Commun Biol
; 6(1): 1160, 2023 11 13.
Artigo
Inglês
| MEDLINE | ID: mdl-37957415
19.
Amino acid residues of both the extracellular and transmembrane domains influence binding of the antiparasitic agent milbemycin to Haemonchus contortus AVR-14B glutamate-gated chloride channels.
Biochem Biophys Res Commun
; 419(3): 562-6, 2012 Mar 16.
Artigo
Inglês
| MEDLINE | ID: mdl-22369940
20.
Competitive antagonism of insect GABA receptors by iminopyridazine derivatives of GABA.
Bioorg Med Chem
; 20(19): 5957-64, 2012 Oct 01.
Artigo
Inglês
| MEDLINE | ID: mdl-22925448