Detalhe da pesquisa
1.
Structure-Based Design, Docking and Binding Free Energy Calculations of A366 Derivatives as Spindlin1 Inhibitors.
Int J Mol Sci
; 22(11)2021 May 31.
Artigo
Inglês
| MEDLINE | ID: mdl-34072837
2.
Comparative Study of the Synthesis and Structural and Physicochemical Properties of Diketopiperazines vs Aza-diketopiperazines.
J Org Chem
; 82(6): 3239-3244, 2017 03 17.
Artigo
Inglês
| MEDLINE | ID: mdl-28230990
3.
Beyond the BET Family: Targeting CBP/p300 with 4-Acyl Pyrroles.
Angew Chem Int Ed Engl
; 56(41): 12476-12480, 2017 10 02.
Artigo
Inglês
| MEDLINE | ID: mdl-28766825
4.
Convenient Access to Fluorescent Probes by Chemoselective Acylation of Hydrazinopeptides: Application to the Synthesis of the First Far-Red Ligand for Apelin Receptor Imaging.
Chemistry
; 22(4): 1399-405, 2016 Jan 22.
Artigo
Inglês
| MEDLINE | ID: mdl-26682530
5.
A step-economical multicomponent synthesis of 3D-shaped aza-diketopiperazines and their drug-like chemical space analysis.
Org Biomol Chem
; 14(37): 8859-8863, 2016 Sep 21.
Artigo
Inglês
| MEDLINE | ID: mdl-27722636
6.
A novel pan-selective bromodomain inhibitor for epigenetic drug design.
Eur J Med Chem
; 249: 115139, 2023 Mar 05.
Artigo
Inglês
| MEDLINE | ID: mdl-36736153
7.
4-Acyl Pyrroles as Dual BET-BRD7/9 Bromodomain Inhibitors Address BETi Insensitive Human Cancer Cell Lines.
J Med Chem
; 63(24): 15603-15620, 2020 12 24.
Artigo
Inglês
| MEDLINE | ID: mdl-33275431
8.
Discovery of a Locally and Orally Active CXCL12 Neutraligand (LIT-927) with Anti-inflammatory Effect in a Murine Model of Allergic Airway Hypereosinophilia.
J Med Chem
; 61(17): 7671-7686, 2018 09 13.
Artigo
Inglês
| MEDLINE | ID: mdl-30106292
9.
Diastereoselective synthesis of novel aza-diketopiperazines via a domino cyclohydrocarbonylation/addition process.
Chem Commun (Camb)
; 50(68): 9657-60, 2014 Sep 04.
Artigo
Inglês
| MEDLINE | ID: mdl-25019687