1.
Bioorg Med Chem Lett
; 16(21): 5567-71, 2006 Nov 01.
Artigo
em Inglês
| MEDLINE
| ID: mdl-16945526
RESUMO
Two series of novel thienopyrrole inhibitors of recombinant human liver glycogen phosphorylase a (GPa) which are effective in reducing glucose output from rat hepatocytes are described. Representative compounds have been shown to bind at the dimer interface site of the rabbit muscle enzyme by X-ray crystallography.