1.
Synthesis and antiproliferative activity of new bioconjugates of Salinomycin with amino acid esters.
Bioorg Med Chem Lett
; 25(17): 3511-4, 2015 Sep 01.
Artigo
em Inglês
| MEDLINE
| ID: mdl-26163197
RESUMO
New Salinomycin (SAL) bioconjugates with amino acid methyl esters were obtained and their antiproliferative activity against cancer cell lines including drug-resistant ones was studied. New compounds exhibit antiproliferative activity towards leukemia and doxorubicin-resistant colon adenocarcinoma cell line and are more effective and less toxic than the commonly currently used anticancer drugs.