Detalhe da pesquisa
1.
Multiplexed cellular profiling identifies an organoselenium compound as an inhibitor of CRM1-mediated nuclear export.
Traffic
; 23(12): 587-599, 2022 12.
Artigo
Inglês
| MEDLINE | ID: mdl-36353954
2.
Boron-containing carbonic anhydrases inhibitors.
Bioorg Chem
; 143: 106976, 2024 Feb.
Artigo
Inglês
| MEDLINE | ID: mdl-38000350
3.
Novel 2-(hydrazinocarbonyl)-3-phenyl-1H-indole-5-sulfonamide based thiosemicarbazides as potent and selective inhibitors of tumor-associated human carbonic anhydrase IX and XII: Synthesis, cytotoxicity, and molecular modelling studies.
Bioorg Chem
; 144: 107096, 2024 Mar.
Artigo
Inglês
| MEDLINE | ID: mdl-38290186
4.
A comparative study of diaryl urea molecules with and without sulfonamide group on Carbonic anhydrase IX and XII inhibition and its consequence on breast cancer cells.
Bioorg Chem
; 145: 107192, 2024 Apr.
Artigo
Inglês
| MEDLINE | ID: mdl-38382393
5.
Identification of thienopyrimidine derivatives tethered with sulfonamide and other moieties as carbonic anhydrase inhibitors: Design, synthesis and anti-proliferative activity.
Bioorg Chem
; 144: 107089, 2024 Mar.
Artigo
Inglês
| MEDLINE | ID: mdl-38237393
6.
Coumarins-lipophilic cations conjugates: Efficient mitocans targeting carbonic anhydrases.
Bioorg Chem
; 145: 107168, 2024 Apr.
Artigo
Inglês
| MEDLINE | ID: mdl-38354500
7.
Synthesis, carbonic anhydrase inhibition studies and modelling investigations of phthalimide-hydantoin hybrids.
J Enzyme Inhib Med Chem
; 39(1): 2335927, 2024 Dec.
Artigo
Inglês
| MEDLINE | ID: mdl-38606915
8.
In-vitro and in-silico investigations of SLC-0111 hydrazinyl analogs as human carbonic anhydrase I, II, IX, and XII inhibitors.
Arch Pharm (Weinheim)
; : e2400157, 2024 May 07.
Artigo
Inglês
| MEDLINE | ID: mdl-38713910
9.
Chemistry of heterocycles as carbonic anhydrase inhibitors: A pathway to novel research in medicinal chemistry review.
Arch Pharm (Weinheim)
; : e2400073, 2024 Apr 29.
Artigo
Inglês
| MEDLINE | ID: mdl-38683875
10.
Sulfonamide-incorporated bis(α-aminophosphonates) as promising carbonic anhydrase inhibitors: Design, synthesis, biological evaluation, and X-ray crystallographic studies.
Arch Pharm (Weinheim)
; : e2400038, 2024 Mar 18.
Artigo
Inglês
| MEDLINE | ID: mdl-38498884
11.
1,2,3-Triazole-based esters and carboxylic acids as nonclassical carbonic anhydrase inhibitors capable of cathepsin B inhibition.
Arch Pharm (Weinheim)
; 357(3): e2300372, 2024 Mar.
Artigo
Inglês
| MEDLINE | ID: mdl-38012535
12.
Exploring rhodanine linked enamine-carbohydrazide derivatives as mycobacterial carbonic anhydrase inhibitors: Design, synthesis, biological evaluation, and molecular docking studies.
Arch Pharm (Weinheim)
; : e2400064, 2024 Mar 18.
Artigo
Inglês
| MEDLINE | ID: mdl-38498883
13.
Design, synthesis, and biological evaluation of 3-benzenesulfonamide-linked 3-hydrazinoisatin derivatives as carbonic anhydrase inhibitors.
Arch Pharm (Weinheim)
; : e2300718, 2024 Mar 11.
Artigo
Inglês
| MEDLINE | ID: mdl-38466120
14.
Identification of 3-(5-cyano-6-oxo-pyridin-2-yl)benzenesulfonamides as novel anticancer agents endowed with EGFR inhibitory activity.
Arch Pharm (Weinheim)
; 357(1): e2300449, 2024 Jan.
Artigo
Inglês
| MEDLINE | ID: mdl-37828544
15.
Novel sulfonamide-phosphonate conjugates as carbonic anhydrase isozymes inhibitors.
Drug Dev Res
; 85(1): e22135, 2024 Feb.
Artigo
Inglês
| MEDLINE | ID: mdl-37997034
16.
Benzothiadiazinone-1,1-Dioxide Carbonic Anhydrase Inhibitors Suppress the Growth of Drug-Resistant Mycobacterium tuberculosis Strains.
Int J Mol Sci
; 25(5)2024 Feb 23.
Artigo
Inglês
| MEDLINE | ID: mdl-38473830
17.
Leveraging SARS-CoV-2 Main Protease (Mpro) for COVID-19 Mitigation with Selenium-Based Inhibitors.
Int J Mol Sci
; 25(2)2024 Jan 12.
Artigo
Inglês
| MEDLINE | ID: mdl-38256046
18.
Mitochondrial carbonic anhydrase VA and VB: properties and roles in health and disease.
J Physiol
; 601(2): 257-274, 2023 01.
Artigo
Inglês
| MEDLINE | ID: mdl-36464834
19.
A simple yet multifaceted 90 years old, evergreen enzyme: Carbonic anhydrase, its inhibition and activation.
Bioorg Med Chem Lett
; 93: 129411, 2023 09 01.
Artigo
Inglês
| MEDLINE | ID: mdl-37507055
20.
Potent and selective carbonic anhydrase inhibition activities of pyrazolones bearing benzenesulfonamides.
Bioorg Med Chem Lett
; 95: 129479, 2023 10 15.
Artigo
Inglês
| MEDLINE | ID: mdl-37704010