Detalhe da pesquisa
1.
Mechanism-specific assay design facilitates the discovery of Nav1.7-selective inhibitors.
Proc Natl Acad Sci U S A
; 115(4): E792-E801, 2018 01 23.
Artigo
Inglês
| MEDLINE | ID: mdl-29311306
2.
Discovery of Acyl-sulfonamide Nav1.7 Inhibitors GDC-0276 and GDC-0310.
J Med Chem
; 64(6): 2953-2966, 2021 03 25.
Artigo
Inglês
| MEDLINE | ID: mdl-33682420
3.
Structural basis of Nav1.7 inhibition by an isoform-selective small-molecule antagonist.
Science
; 350(6267): aac5464, 2015 Dec 18.
Artigo
Inglês
| MEDLINE | ID: mdl-26680203
4.
Treatment of Na(v)1.7-mediated pain in inherited erythromelalgia using a novel sodium channel blocker.
Pain
; 153(1): 80-85, 2012 Jan.
Artigo
Inglês
| MEDLINE | ID: mdl-22035805