Detalhe da pesquisa
1.
Benzimidazole-based DGAT1 inhibitors with a [3.1.0] bicyclohexane carboxylic acid moiety.
Bioorg Med Chem Lett
; 29(10): 1182-1186, 2019 05 15.
Artigo
Inglês
| MEDLINE | ID: mdl-30926247
2.
Constraining the amide bond in N-sulfonylated dipeptide VLA-4 antagonists.
Bioorg Med Chem Lett
; 18(5): 1688-91, 2008 Mar 01.
Artigo
Inglês
| MEDLINE | ID: mdl-18242984
3.
Discovery of a Potent and Selective DGAT1 Inhibitor with a Piperidinyl-oxy-cyclohexanecarboxylic Acid Moiety.
ACS Med Chem Lett
; 5(10): 1082-7, 2014 Oct 09.
Artigo
Inglês
| MEDLINE | ID: mdl-25349648
4.
Potent DGAT1 Inhibitors in the Benzimidazole Class with a Pyridyl-oxy-cyclohexanecarboxylic Acid Moiety.
ACS Med Chem Lett
; 4(8): 773-8, 2013 Aug 08.
Artigo
Inglês
| MEDLINE | ID: mdl-24900745
5.
VLA-4 antagonists: potent inhibitors of lymphocyte migration.
Med Res Rev
; 23(3): 369-92, 2003 May.
Artigo
Inglês
| MEDLINE | ID: mdl-12647315
6.
Substituted tetrahydrofuroyl-1-phenylalanine derivatives as potent and specific VLA-4 antagonists.
Bioorg Med Chem Lett
; 12(11): 1501-5, 2002 Jun 03.
Artigo
Inglês
| MEDLINE | ID: mdl-12031329
7.
N-isonicotinoyl-(L)-4-aminophenylalanine derivatives as tight binding VLA-4 antagonists.
Bioorg Med Chem Lett
; 13(11): 1891-5, 2003 Jun 02.
Artigo
Inglês
| MEDLINE | ID: mdl-12749892
8.
N-Tetrahydrofuroyl-(L)-phenylalanine derivatives as potent VLA-4 antagonists.
Bioorg Med Chem Lett
; 12(11): 1497-500, 2002 Jun 03.
Artigo
Inglês
| MEDLINE | ID: mdl-12031328