Detalhe da pesquisa
1.
Genomic and virulence analysis of in vitro cultured Cryptosporidium parvum.
PLoS Pathog
; 20(2): e1011992, 2024 Feb.
Artigo
Inglês
| MEDLINE | ID: mdl-38416794
2.
P-Glycoprotein-Mediated Efflux Reduces the In Vivo Efficacy of a Therapeutic Targeting the Gastrointestinal Parasite Cryptosporidium.
J Infect Dis
; 220(7): 1188-1198, 2019 08 30.
Artigo
Inglês
| MEDLINE | ID: mdl-31180118
3.
Assessment of a pretomanid analogue library for African trypanosomiasis: Hit-to-lead studies on 6-substituted 2-nitro-6,7-dihydro-5H-imidazo[2,1-b][1,3]thiazine 8-oxides.
Bioorg Med Chem Lett
; 28(2): 207-213, 2018 01 15.
Artigo
Inglês
| MEDLINE | ID: mdl-29191556
4.
Eicosapentaenoic Acid Modulates Trichomonas vaginalis Activity.
J Eukaryot Microbiol
; 63(2): 153-61, 2016.
Artigo
Inglês
| MEDLINE | ID: mdl-26333486
5.
Cryptosporidium parvum induces an endoplasmic stress response in the intestinal adenocarcinoma HCT-8 cell line.
J Biol Chem
; 288(42): 30356-30364, 2013 Oct 18.
Artigo
Inglês
| MEDLINE | ID: mdl-23986438
6.
Pharmacokinetics and pharmacodynamics utilizing unbound target tissue exposure as part of a disposition-based rationale for lead optimization of benzoxaboroles in the treatment of Stage 2 Human African Trypanosomiasis.
Parasitology
; 141(1): 104-18, 2014 Jan.
Artigo
Inglês
| MEDLINE | ID: mdl-24007596
7.
SAR of 2-amino and 2,4-diamino pyrimidines with in vivo efficacy against Trypanosoma brucei.
Bioorg Med Chem Lett
; 21(10): 2816-9, 2011 May 15.
Artigo
Inglês
| MEDLINE | ID: mdl-21507639
8.
Bis(oxyphenylene)benzimidazoles: a novel class of anti-Plasmodium falciparum agents.
Bioorg Med Chem
; 19(24): 7493-500, 2011 Dec 15.
Artigo
Inglês
| MEDLINE | ID: mdl-22061825
9.
Oxygen levels are key to understanding "Anaerobic" protozoan pathogens with micro-aerophilic lifestyles.
Adv Microb Physiol
; 79: 163-240, 2021.
Artigo
Inglês
| MEDLINE | ID: mdl-34836611
10.
Discovery of novel orally bioavailable oxaborole 6-carboxamides that demonstrate cure in a murine model of late-stage central nervous system african trypanosomiasis.
Antimicrob Agents Chemother
; 54(10): 4379-88, 2010 Oct.
Artigo
Inglês
| MEDLINE | ID: mdl-20660666
11.
Arginine metabolism in Trichomonas vaginalis infected with Mycoplasma hominis.
Microbiology (Reading)
; 156(Pt 12): 3734-3743, 2010 Dec.
Artigo
Inglês
| MEDLINE | ID: mdl-20656780
12.
In Vitro Culture of Cryptosporidium parvum Using Hollow Fiber Bioreactor: Applications for Simultaneous Pharmacokinetic and Pharmacodynamic Evaluation of Test Compounds.
Methods Mol Biol
; 2052: 335-350, 2020.
Artigo
Inglês
| MEDLINE | ID: mdl-31452171
13.
Metabolism of an alkyl polyamine analog by a polyamine oxidase from the microsporidian Encephalitozoon cuniculi.
Antimicrob Agents Chemother
; 53(6): 2599-604, 2009 Jun.
Artigo
Inglês
| MEDLINE | ID: mdl-19223636
14.
Trypanocidal activity of 8-methyl-5'-{[(Z)-4-aminobut-2-enyl]-(methylamino)}adenosine (Genz-644131), an adenosylmethionine decarboxylase inhibitor.
Antimicrob Agents Chemother
; 53(8): 3269-72, 2009 Aug.
Artigo
Inglês
| MEDLINE | ID: mdl-19451291
15.
Novel S-adenosylmethionine decarboxylase inhibitors for the treatment of human African trypanosomiasis.
Antimicrob Agents Chemother
; 53(5): 2052-8, 2009 May.
Artigo
Inglês
| MEDLINE | ID: mdl-19289530
16.
Synthesis and SAR of alkanediamide-linked bisbenzamidines with anti-trypanosomal and anti-pneumocystis activity.
Bioorg Med Chem Lett
; 19(20): 5884-6, 2009 Oct 15.
Artigo
Inglês
| MEDLINE | ID: mdl-19736009
17.
Novel Synthetic Polyamines Have Potent Antimalarial Activities in vitro and in vivo by Decreasing Intracellular Spermidine and Spermine Concentrations.
Front Cell Infect Microbiol
; 9: 9, 2019.
Artigo
Inglês
| MEDLINE | ID: mdl-30838177
18.
Long-term in vitro Culture of Cryptosporidium parvum.
Bio Protoc
; 8(15): e2947, 2018 Aug 05.
Artigo
Inglês
| MEDLINE | ID: mdl-34395759
19.
Mitochondrial Glycolysis in a Major Lineage of Eukaryotes.
Genome Biol Evol
; 10(9): 2310-2325, 2018 09 01.
Artigo
Inglês
| MEDLINE | ID: mdl-30060189
20.
Cryptosporidium parvum spermidine/spermine N1-acetyltransferase exhibits different characteristics from the host enzyme.
Mol Biochem Parasitol
; 152(2): 170-80, 2007 Apr.
Artigo
Inglês
| MEDLINE | ID: mdl-17289169