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The preclinical efficacy, selectivity and pharmacologic profile of MK-5932, an insulin-sparing selective glucocorticoid receptor modulator.
Brandish, Philip E; Anderson, Kenneth; Baltus, Gretchen A; Bai, Chang; Bungard, Christopher J; Bunting, Patricia; Byford, Alan; Chiu, Chi-Sung; Cicmil, Milenko; Corcoran, Halea; Euler, Danielle; Fisher, John E; Gambone, Carlo; Hasbun-Manning, Martha; Kuklin, Nelly; Landis, Elizabeth; Lifsted, Traci Q; McElwee-Witmer, Sheila; McIntosh, Ian S; Meissner, Robert S; Miao, John; Mitchell, Helen J; Musselman, Amy; Schmidt, Azriel; Shin, John; Szczerba, Peter; Thompson, Charles D; Tribouley, Catherine; Vogel, Robert L; Warrier, Sudha; Hershey, James C.
  • Brandish PE; Merck & Co., Inc., Boston, MA 02115, United States. Electronic address: philip.brandish@merck.com.
  • Anderson K; Merck & Co., Inc., West Point, PA 19422, United States.
  • Baltus GA; Merck & Co., Inc., Boston, MA 02115, United States.
  • Bai C; Merck & Co., Inc., West Point, PA 19422, United States.
  • Bungard CJ; Merck & Co., Inc., West Point, PA 19422, United States.
  • Bunting P; Merck & Co., Inc., West Point, PA 19422, United States.
  • Byford A; Merck & Co., Inc., Boston, MA 02115, United States.
  • Chiu CS; Merck & Co., Inc., Boston, MA 02115, United States.
  • Cicmil M; Merck & Co., Inc., Boston, MA 02115, United States.
  • Corcoran H; Merck & Co., Inc., West Point, PA 19422, United States.
  • Euler D; Merck & Co., Inc., West Point, PA 19422, United States.
  • Fisher JE; Merck & Co., Inc., West Point, PA 19422, United States.
  • Gambone C; Merck & Co., Inc., West Point, PA 19422, United States.
  • Hasbun-Manning M; Merck & Co., Inc., West Point, PA 19422, United States.
  • Kuklin N; Merck & Co., Inc., Boston, MA 02115, United States.
  • Landis E; Merck & Co., Inc., West Point, PA 19422, United States.
  • Lifsted TQ; Merck & Co., Inc., West Point, PA 19422, United States.
  • McElwee-Witmer S; Merck & Co., Inc., West Point, PA 19422, United States.
  • McIntosh IS; Merck & Co., Inc., West Point, PA 19422, United States.
  • Meissner RS; Merck & Co., Inc., West Point, PA 19422, United States.
  • Miao J; Merck & Co., Inc., Boston, MA 02115, United States.
  • Mitchell HJ; Merck & Co., Inc., West Point, PA 19422, United States.
  • Musselman A; Merck & Co., Inc., West Point, PA 19422, United States.
  • Schmidt A; Merck & Co., Inc., West Point, PA 19422, United States.
  • Shin J; Merck & Co., Inc., Boston, MA 02115, United States.
  • Szczerba P; Merck & Co., Inc., West Point, PA 19422, United States.
  • Thompson CD; Merck & Co., Inc., West Point, PA 19422, United States.
  • Tribouley C; Merck & Co., Inc., Boston, MA 02115, United States.
  • Vogel RL; Merck & Co., Inc., West Point, PA 19422, United States.
  • Warrier S; Merck & Co., Inc., West Point, PA 19422, United States.
  • Hershey JC; Merck & Co., Inc., West Point, PA 19422, United States.
Eur J Pharmacol ; 724: 102-11, 2014 Feb 05.
Article en En | MEDLINE | ID: mdl-24374007

Texto completo: 1 Banco de datos: MEDLINE Asunto principal: Artritis Experimental / Benzamidas / Receptores de Glucocorticoides / Dermatitis por Contacto / Edema / Indazoles / Antiinflamatorios Límite: Animals / Female / Humans / Male Idioma: En Año: 2014 Tipo del documento: Article

Texto completo: 1 Banco de datos: MEDLINE Asunto principal: Artritis Experimental / Benzamidas / Receptores de Glucocorticoides / Dermatitis por Contacto / Edema / Indazoles / Antiinflamatorios Límite: Animals / Female / Humans / Male Idioma: En Año: 2014 Tipo del documento: Article