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Development and characterisation of novel fentanyl-delta opioid receptor antagonist based bivalent ligands.
Bird, M F; Vardanyan, R S; Hruby, V J; Calò, G; Guerrini, R; Salvadori, S; Trapella, C; McDonald, J; Rowbotham, D J; Lambert, D G.
  • Bird MF; Department of Cardiovascular Sciences, Division of Anaesthesia, Critical Care and Pain Management, University of Leicester, Robert Kilpatrick Clinical Sciences Building, Leicester Royal Infirmary, Leicester LE2 7LX, UK.
  • Vardanyan RS; Department of Chemistry and Biochemistry, University of Arizona, Tucson, AZ 85721, USA.
  • Hruby VJ; Department of Chemistry and Biochemistry, University of Arizona, Tucson, AZ 85721, USA.
  • Calò G; Department of Medical Sciences, Section of Pharmacology, University of Ferrara and Italian Institute of Neuroscience, Ferrara, Italy.
  • Guerrini R; Department of Chemical and Pharmaceutical Sciences and LTTA (Laboratorio per le Tecnologie delle Terapie Avanzate), University of Ferrara, Ferrara, Italy.
  • Salvadori S; Department of Chemical and Pharmaceutical Sciences and LTTA (Laboratorio per le Tecnologie delle Terapie Avanzate), University of Ferrara, Ferrara, Italy.
  • Trapella C; Department of Chemical and Pharmaceutical Sciences and LTTA (Laboratorio per le Tecnologie delle Terapie Avanzate), University of Ferrara, Ferrara, Italy.
  • McDonald J; Department of Cardiovascular Sciences, Division of Anaesthesia, Critical Care and Pain Management, University of Leicester, Robert Kilpatrick Clinical Sciences Building, Leicester Royal Infirmary, Leicester LE2 7LX, UK.
  • Rowbotham DJ; Department of Cardiovascular Sciences, Division of Anaesthesia, Critical Care and Pain Management, University of Leicester, Robert Kilpatrick Clinical Sciences Building, Leicester Royal Infirmary, Leicester LE2 7LX, UK.
  • Lambert DG; Department of Cardiovascular Sciences, Division of Anaesthesia, Critical Care and Pain Management, University of Leicester, Robert Kilpatrick Clinical Sciences Building, Leicester Royal Infirmary, Leicester LE2 7LX, UK dgl3@le.ac.uk.
Br J Anaesth ; 114(4): 646-56, 2015 Apr.
Article en En | MEDLINE | ID: mdl-25680364

Texto completo: 1 Banco de datos: MEDLINE Asunto principal: Fentanilo / Receptores Opioides delta / Tetrahidroisoquinolinas / Dipéptidos Límite: Animals Idioma: En Año: 2015 Tipo del documento: Article

Texto completo: 1 Banco de datos: MEDLINE Asunto principal: Fentanilo / Receptores Opioides delta / Tetrahidroisoquinolinas / Dipéptidos Límite: Animals Idioma: En Año: 2015 Tipo del documento: Article