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Crystal structures of the M1 and M4 muscarinic acetylcholine receptors.
Thal, David M; Sun, Bingfa; Feng, Dan; Nawaratne, Vindhya; Leach, Katie; Felder, Christian C; Bures, Mark G; Evans, David A; Weis, William I; Bachhawat, Priti; Kobilka, Tong Sun; Sexton, Patrick M; Kobilka, Brian K; Christopoulos, Arthur.
  • Thal DM; Drug Discovery Biology and Department of Pharmacology, Monash Institute of Pharmaceutical Sciences, Monash University, Parkville, 3052, Victoria, Australia.
  • Sun B; ConfometRx, 3070 Kenneth Street, Santa Clara, California 95054, USA.
  • Feng D; ConfometRx, 3070 Kenneth Street, Santa Clara, California 95054, USA.
  • Nawaratne V; Drug Discovery Biology and Department of Pharmacology, Monash Institute of Pharmaceutical Sciences, Monash University, Parkville, 3052, Victoria, Australia.
  • Leach K; Drug Discovery Biology and Department of Pharmacology, Monash Institute of Pharmaceutical Sciences, Monash University, Parkville, 3052, Victoria, Australia.
  • Felder CC; Neuroscience, Eli Lilly, Indianapolis, Indiana 46285, USA.
  • Bures MG; Computational Chemistry and Chemoinformatics, Eli Lilly, Indianapolis, Indiana 46285, USA.
  • Evans DA; Computational Chemistry and Chemoinformatics, Eli Lilly, Sunninghill Road, Windlesham GU20 6PH, UK.
  • Weis WI; Department of Molecular and Cellular Physiology, Stanford University School of Medicine, Stanford, California 94305, USA.
  • Bachhawat P; Department of Structural Biology, Stanford University School of Medicine, Stanford, California 94305, USA.
  • Kobilka TS; ConfometRx, 3070 Kenneth Street, Santa Clara, California 95054, USA.
  • Sexton PM; ConfometRx, 3070 Kenneth Street, Santa Clara, California 95054, USA.
  • Kobilka BK; Drug Discovery Biology and Department of Pharmacology, Monash Institute of Pharmaceutical Sciences, Monash University, Parkville, 3052, Victoria, Australia.
  • Christopoulos A; ConfometRx, 3070 Kenneth Street, Santa Clara, California 95054, USA.
Nature ; 531(7594): 335-40, 2016 Mar 17.
Article en En | MEDLINE | ID: mdl-26958838

Texto completo: 1 Banco de datos: MEDLINE Asunto principal: Receptor Muscarínico M1 / Receptor Muscarínico M4 Límite: Humans Idioma: En Año: 2016 Tipo del documento: Article

Texto completo: 1 Banco de datos: MEDLINE Asunto principal: Receptor Muscarínico M1 / Receptor Muscarínico M4 Límite: Humans Idioma: En Año: 2016 Tipo del documento: Article