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Time-dependent inhibition of PHD2.
Tcholakov, Isabelle; Grimshaw, Charles E; Shi, Lihong; Kiryanov, Andre; Murphy, Sean T; Larson, Christopher J; Plonowski, Artur; Ermolieff, Jacques.
  • Tcholakov I; In Vitro Pharmacology, Immunology, Takeda California, Inc., 10410 Science Center Drive, San Diego, CA 92121, U.S.A.
  • Grimshaw CE; Enzymology and Biophysical Chemistry, Takeda California, Inc., 10410 Science Center Drive, San Diego, CA 92121, U.S.A.
  • Shi L; Enzymology and Biophysical Chemistry, Takeda California, Inc., 10410 Science Center Drive, San Diego, CA 92121, U.S.A.
  • Kiryanov A; Medicinal Chemistry, Takeda California, Inc., 10410 Science Center Drive, San Diego, CA 92121, U.S.A.
  • Murphy ST; Medicinal Chemistry, Takeda California, Inc., 10410 Science Center Drive, San Diego, CA 92121, U.S.A.
  • Larson CJ; External Innovation, Takeda California, Inc., 10410 Science Center Drive, San Diego, CA 92121, U.S.A.
  • Plonowski A; Metabolic Disease, Takeda California, Inc., 10410 Science Center Drive, San Diego, CA 92121, U.S.A.
  • Ermolieff J; In Vitro Pharmacology, Gastrointestinal and Enterology Discovery Unit, Takeda California, Inc., 10410 Science Center Drive, San Diego, CA 92121, U.S.A. jacques.ermolieff@takeda.com.
Biosci Rep ; 37(3)2017 Jun 30.
Article en En | MEDLINE | ID: mdl-28592559

Texto completo: 1 Banco de datos: MEDLINE Asunto principal: Inhibidores Enzimáticos / Bibliotecas de Moléculas Pequeñas / Prolina Dioxigenasas del Factor Inducible por Hipoxia Límite: Humans Idioma: En Año: 2017 Tipo del documento: Article

Texto completo: 1 Banco de datos: MEDLINE Asunto principal: Inhibidores Enzimáticos / Bibliotecas de Moléculas Pequeñas / Prolina Dioxigenasas del Factor Inducible por Hipoxia Límite: Humans Idioma: En Año: 2017 Tipo del documento: Article