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Targeted Blockade of TARP-γ8-Associated AMPA Receptors: Anticonvulsant Activity with the Selective Antagonist LY3130481 (CERC-611).
Witkin, Jeffrey M; Schober, Douglas A; Gleason, Scott D; Catlow, John T; Porter, Warren J; Reel, Jon; Jin, Xiaoming; Hobbs, Jonathan; Gehlert, Donald; Gernert, Douglas L; Gardinier, Kevin M; Kato, Akihiko S; Ping, Xingjie; Smith, Jodi L.
  • Witkin JM; Lilly Research Laboratories, Eli Lilly and Company, Indianapolis, Indiana, United States.
  • Schober DA; Lilly Research Laboratories, Eli Lilly and Company, Indianapolis, Indiana, United States.
  • Gleason SD; Lilly Research Laboratories, Eli Lilly and Company, Indianapolis, Indiana, United States.
  • Catlow JT; Lilly Research Laboratories, Eli Lilly and Company, Indianapolis, Indiana, United States.
  • Porter WJ; Lilly Research Laboratories, Eli Lilly and Company, Indianapolis, Indiana, United States.
  • Reel J; Lilly Research Laboratories, Eli Lilly and Company, Indianapolis, Indiana, United States.
  • Jin X; Indiana University/Purdue University, Riley Hospital, Indianapolis, Indiana, United States.
  • Hobbs J; Indiana University/Purdue University, Riley Hospital, Indianapolis, Indiana, United States.
  • Gehlert D; Cerecor, Baltimore, MD (DG) and Matrix Pharmaceutical Consulting, Boulder, CO, United States.
  • Gernert DL; Lilly Research Laboratories, Eli Lilly and Company, Indianapolis, Indiana, United States.
  • Gardinier KM; Lilly Research Laboratories, Eli Lilly and Company, Indianapolis, Indiana, United States.
  • Kato AS; Lilly Research Laboratories, Eli Lilly and Company, Indianapolis, Indiana, United States.
  • Ping X; Indiana University/Purdue University, Riley Hospital, Indianapolis, Indiana, United States.
  • Smith JL; Indiana University/Purdue University, Riley Hospital, Indianapolis, Indiana, United States.
CNS Neurol Disord Drug Targets ; 16(10): 1099-1110, 2017.
Article en En | MEDLINE | ID: mdl-29090671

Texto completo: 1 Banco de datos: MEDLINE Asunto principal: Pirazoles / Convulsiones / Canales de Calcio / Receptores AMPA / Benzotiazoles Tipo de estudio: Prognostic_studies / Risk_factors_studies Límite: Animals / Female / Humans / Male Idioma: En Año: 2017 Tipo del documento: Article

Texto completo: 1 Banco de datos: MEDLINE Asunto principal: Pirazoles / Convulsiones / Canales de Calcio / Receptores AMPA / Benzotiazoles Tipo de estudio: Prognostic_studies / Risk_factors_studies Límite: Animals / Female / Humans / Male Idioma: En Año: 2017 Tipo del documento: Article