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Discovery of an Irreversible and Cell-Active BCL6 Inhibitor Selectively Targeting Cys53 Located at the Protein-Protein Interaction Interface.
Sameshima, Tomoya; Yamamoto, Takeshi; Sano, Osamu; Sogabe, Satoshi; Igaki, Shigeru; Sakamoto, Kotaro; Ida, Koh; Gotou, Mika; Imaeda, Yasuhiro; Sakamoto, Junichi; Miyahisa, Ikuo.
  • Sameshima T; Pharmaceutical Research Division, Takeda Pharmaceutical Company Limited , 26-1, Muraoka-higashi 2 chome, Fujisawa, Kanagawa 251-8555, Japan.
  • Yamamoto T; Pharmaceutical Research Division, Takeda Pharmaceutical Company Limited , 26-1, Muraoka-higashi 2 chome, Fujisawa, Kanagawa 251-8555, Japan.
  • Sano O; Pharmaceutical Research Division, Takeda Pharmaceutical Company Limited , 26-1, Muraoka-higashi 2 chome, Fujisawa, Kanagawa 251-8555, Japan.
  • Sogabe S; Pharmaceutical Research Division, Takeda Pharmaceutical Company Limited , 26-1, Muraoka-higashi 2 chome, Fujisawa, Kanagawa 251-8555, Japan.
  • Igaki S; Pharmaceutical Research Division, Takeda Pharmaceutical Company Limited , 26-1, Muraoka-higashi 2 chome, Fujisawa, Kanagawa 251-8555, Japan.
  • Sakamoto K; Pharmaceutical Research Division, Takeda Pharmaceutical Company Limited , 26-1, Muraoka-higashi 2 chome, Fujisawa, Kanagawa 251-8555, Japan.
  • Ida K; Pharmaceutical Research Division, Takeda Pharmaceutical Company Limited , 26-1, Muraoka-higashi 2 chome, Fujisawa, Kanagawa 251-8555, Japan.
  • Gotou M; Pharmaceutical Research Division, Takeda Pharmaceutical Company Limited , 26-1, Muraoka-higashi 2 chome, Fujisawa, Kanagawa 251-8555, Japan.
  • Imaeda Y; Pharmaceutical Research Division, Takeda Pharmaceutical Company Limited , 26-1, Muraoka-higashi 2 chome, Fujisawa, Kanagawa 251-8555, Japan.
  • Sakamoto J; Pharmaceutical Research Division, Takeda Pharmaceutical Company Limited , 26-1, Muraoka-higashi 2 chome, Fujisawa, Kanagawa 251-8555, Japan.
  • Miyahisa I; Pharmaceutical Research Division, Takeda Pharmaceutical Company Limited , 26-1, Muraoka-higashi 2 chome, Fujisawa, Kanagawa 251-8555, Japan.
Biochemistry ; 57(8): 1369-1379, 2018 02 27.
Article en En | MEDLINE | ID: mdl-29293322

Texto completo: 1 Banco de datos: MEDLINE Asunto principal: Proteínas Proto-Oncogénicas c-bcl-6 / Bibliotecas de Moléculas Pequeñas / Mapas de Interacción de Proteínas Límite: Humans Idioma: En Año: 2018 Tipo del documento: Article

Texto completo: 1 Banco de datos: MEDLINE Asunto principal: Proteínas Proto-Oncogénicas c-bcl-6 / Bibliotecas de Moléculas Pequeñas / Mapas de Interacción de Proteínas Límite: Humans Idioma: En Año: 2018 Tipo del documento: Article