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Synthesis and evaluation of a ring-constrained Hsp90 C-terminal inhibitor that exhibits neuroprotective activity.
Zhang, Zheng; You, Zhenyuan; Dobrowsky, Rick T; Blagg, Brian S J.
  • Zhang Z; Department of Chemistry and Biochemistry, The University of Notre Dame, 251 Nieuwland Science Hall, Notre Dame, IN 46556, United States.
  • You Z; Department of Pharmacology and Toxicology Department, The University of Kansas, Lawrence, KS 66045, United States.
  • Dobrowsky RT; Department of Pharmacology and Toxicology Department, The University of Kansas, Lawrence, KS 66045, United States.
  • Blagg BSJ; Department of Chemistry and Biochemistry, The University of Notre Dame, 251 Nieuwland Science Hall, Notre Dame, IN 46556, United States. Electronic address: bblagg@nd.edu.
Bioorg Med Chem Lett ; 28(16): 2701-2704, 2018 09 01.
Article en En | MEDLINE | ID: mdl-29759728

Texto completo: 1 Banco de datos: MEDLINE Asunto principal: Fenantridinas / Fármacos Neuroprotectores / Proteínas HSP90 de Choque Térmico / Glicósidos / Lactamas Límite: Animals Idioma: En Año: 2018 Tipo del documento: Article

Texto completo: 1 Banco de datos: MEDLINE Asunto principal: Fenantridinas / Fármacos Neuroprotectores / Proteínas HSP90 de Choque Térmico / Glicósidos / Lactamas Límite: Animals Idioma: En Año: 2018 Tipo del documento: Article