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Structure-based drug design, synthesis, In vitro, and In vivo biological evaluation of indole-based biomimetic analogs targeting estrogen receptor-α inhibition.
Hendy, Moataz S; Ali, Aya A; Ahmed, Lubna; Hossam, Reham; Mostafa, Alaa; Elmazar, Mohamed M; Naguib, Bassem H; Attia, Yasmeen M; Ahmed, Mahmoud Salama.
  • Hendy MS; Department of Pharmaceutical Chemistry, Faculty of Pharmacy, The British University in Egypt, El-Sherouk, Cairo, Egypt; Center of Drug Research and Development (CDRD), The British University in Egypt, El-Sherouk, Cairo, Egypt.
  • Ali AA; Center of Drug Research and Development (CDRD), The British University in Egypt, El-Sherouk, Cairo, Egypt; Department of Pharmacology, Faculty of Pharmacy, The British University in Egypt, El-Sherouk, Cairo, Egypt.
  • Ahmed L; Faculty of Pharmacy, The British University in Egypt, El-Sherouk, Cairo, Egypt.
  • Hossam R; Faculty of Pharmacy, The British University in Egypt, El-Sherouk, Cairo, Egypt.
  • Mostafa A; Faculty of Pharmacy, The British University in Egypt, El-Sherouk, Cairo, Egypt.
  • Elmazar MM; Center of Drug Research and Development (CDRD), The British University in Egypt, El-Sherouk, Cairo, Egypt; Department of Pharmacology, Faculty of Pharmacy, The British University in Egypt, El-Sherouk, Cairo, Egypt.
  • Naguib BH; Department of Pharmaceutical Chemistry, Faculty of Pharmacy, The British University in Egypt, El-Sherouk, Cairo, Egypt; Center of Drug Research and Development (CDRD), The British University in Egypt, El-Sherouk, Cairo, Egypt; Department of Pharmaceutical Organic Chemistry, Faculty of Pharmacy, Cair
  • Attia YM; Center of Drug Research and Development (CDRD), The British University in Egypt, El-Sherouk, Cairo, Egypt; Department of Pharmacology, Faculty of Pharmacy, The British University in Egypt, El-Sherouk, Cairo, Egypt. Electronic address: Yasmeen.attia@bue.edu.eg.
  • Ahmed MS; Department of Pharmaceutical Chemistry, Faculty of Pharmacy, The British University in Egypt, El-Sherouk, Cairo, Egypt; Center of Drug Research and Development (CDRD), The British University in Egypt, El-Sherouk, Cairo, Egypt; Department of Internal Medicine, Division of Cardiology, University of Te
Eur J Med Chem ; 166: 281-290, 2019 Mar 15.
Article en En | MEDLINE | ID: mdl-30731397

Texto completo: 1 Banco de datos: MEDLINE Asunto principal: Diseño de Fármacos / Materiales Biomiméticos / Receptor alfa de Estrógeno / Indoles / Antineoplásicos Límite: Humans Idioma: En Año: 2019 Tipo del documento: Article

Texto completo: 1 Banco de datos: MEDLINE Asunto principal: Diseño de Fármacos / Materiales Biomiméticos / Receptor alfa de Estrógeno / Indoles / Antineoplásicos Límite: Humans Idioma: En Año: 2019 Tipo del documento: Article