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Synthesis and evaluation of in vivo anti-hypothermic effect of all stereoisomers of the thyrotropin-releasing hormone mimetic: Rovatirelin Hydrate.
Kobayashi, Naotake; Sato, Norihito; Sugita, Katsuji; Takahashi, Kouji; Sugawara, Tamio; Tada, Yukio; Yoshikawa, Takayoshi.
  • Kobayashi N; Medicinal chemistry research laboratory, Shionogi & Co., Ltd. 3-1-1, Futaba-cho, Toyonaka-shi, Osaka, 561-0825, Japan.
  • Sato N; Research Laboratory for Development, Shionogi & Co., Ltd. 3-1-1, Futaba-cho, Toyonaka-shi, Osaka, 561-0825, Japan.
  • Sugita K; Research Laboratory for Development, Shionogi & Co., Ltd. 3-1-1, Futaba-cho, Toyonaka-shi, Osaka, 561-0825, Japan.
  • Takahashi K; DMPK Services, Shionogi Techno Advance Research Co., Ltd. 3-1-1, Futaba-cho, Toyonaka-shi, Osaka, 561-0825, Japan.
  • Sugawara T; Medicinal chemistry research laboratory, Shionogi & Co., Ltd. 3-1-1, Futaba-cho, Toyonaka-shi, Osaka, 561-0825, Japan.
  • Tada Y; Medicinal chemistry research laboratory, Shionogi & Co., Ltd. 3-1-1, Futaba-cho, Toyonaka-shi, Osaka, 561-0825, Japan.
  • Yoshikawa T; Pharmacovigilance Japan, Allergan Japan K.K., 4-20-3-35, Ebisu Shibuya-ku, Tokyo, 150-6035, Japan.
J Pept Sci ; 25(12): e3228, 2019 Dec.
Article en En | MEDLINE | ID: mdl-31713944

Texto completo: 1 Banco de datos: MEDLINE Asunto principal: Pirrolidinas / Oxazolidinonas / Hipotermia Límite: Animals Idioma: En Año: 2019 Tipo del documento: Article

Texto completo: 1 Banco de datos: MEDLINE Asunto principal: Pirrolidinas / Oxazolidinonas / Hipotermia Límite: Animals Idioma: En Año: 2019 Tipo del documento: Article