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Crystal structure of pathogenic Staphylococcus aureus lipase complex with the anti-obesity drug orlistat.
Kitadokoro, Kengo; Tanaka, Mutsumi; Hikima, Takaaki; Okuno, Yukiko; Yamamoto, Masaki; Kamitani, Shigeki.
  • Kitadokoro K; Faculty of Molecular Chemistry and Engineering, Graduate School of Science and Technology, Kyoto Institute of Technology, Hashigami-cho, Matsugasaki, Sakyo-ku, Kyoto, 606-8585, Japan. kengo@kit.ac.jp.
  • Tanaka M; Faculty of Molecular Chemistry and Engineering, Graduate School of Science and Technology, Kyoto Institute of Technology, Hashigami-cho, Matsugasaki, Sakyo-ku, Kyoto, 606-8585, Japan.
  • Hikima T; SR Life Science Instrumentation Team, Life Science Research Infrastructure Group, Advanced Photon Technology Division, RIKEN SPring-8 Center, 1-1-1, Koto, Sayo-cho, Sayo-gun, Hyogo, 679-6148, Japan.
  • Okuno Y; Medical Research Support Center, Graduate School of Medicine, Kyoto University, Yoshidakonoe, Sakyo-ku, Kyoto, 606-8501, Japan.
  • Yamamoto M; SR Life Science Instrumentation Team, Life Science Research Infrastructure Group, Advanced Photon Technology Division, RIKEN SPring-8 Center, 1-1-1, Koto, Sayo-cho, Sayo-gun, Hyogo, 679-6148, Japan.
  • Kamitani S; Graduate School of Comprehensive Rehabilitation, College of Health and Human Sciences, Osaka Prefecture University, 3-7-30 Habikino, Habikino, 583-8555, Osaka, Japan.
Sci Rep ; 10(1): 5469, 2020 03 25.
Article en En | MEDLINE | ID: mdl-32214208

Texto completo: 1 Banco de datos: MEDLINE Asunto principal: Staphylococcus aureus / Fármacos Antiobesidad / Factores de Virulencia / Inhibidores Enzimáticos / Esterasas / Reposicionamiento de Medicamentos / Desarrollo de Medicamentos / Orlistat / Antibacterianos Tipo de estudio: Prognostic_studies Idioma: En Año: 2020 Tipo del documento: Article

Texto completo: 1 Banco de datos: MEDLINE Asunto principal: Staphylococcus aureus / Fármacos Antiobesidad / Factores de Virulencia / Inhibidores Enzimáticos / Esterasas / Reposicionamiento de Medicamentos / Desarrollo de Medicamentos / Orlistat / Antibacterianos Tipo de estudio: Prognostic_studies Idioma: En Año: 2020 Tipo del documento: Article