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Azetidine-based selective glycine transporter-1 (GlyT1) inhibitors with memory enhancing properties.
Hudson, Andrew R; Santora, Vincent J; Petroski, Robert E; Almos, Theresa A; Anderson, Gary; Barido, Richard; Basinger, Jillian; Bellows, Chris L; Bookser, Brett C; Broadbent, Nicola J; Cabebe, Clifford; Chai, Chih-Kun; Chen, Mi; Chow, Stephine; Chung, De Michael; Heger, Lindsay; Danks, Anne M; Freestone, Graeme C; Gitnick, Dany; Gupta, Varsha; Hoffmaster, Christine; Kaplan, Alan P; Kennedy, Michael R; Lee, Dong; Limberis, James; Ly, Kiev; Mak, Chi Ching; Masatsugu, Brittany; Morse, Andrew C; Na, Jim; Neul, David; Nikpur, John; Renick, Joel; Sebring, Kristen; Sevidal, Samantha; Tabatabaei, Ali; Wen, Jenny; Xia, Shouzhen; Yan, Yingzhuo; Yoder, Zachary W; Zook, Douglas; Peters, Marco; Breitenbucher, J Guy.
  • Hudson AR; Dart Neuroscience, 12278 Scripps Summit Dr, San Diego, CA 92131, United States. Electronic address: andyrhudson@gmail.com.
  • Santora VJ; Dart Neuroscience, 12278 Scripps Summit Dr, San Diego, CA 92131, United States.
  • Petroski RE; Dart Neuroscience, 12278 Scripps Summit Dr, San Diego, CA 92131, United States.
  • Almos TA; Dart Neuroscience, 12278 Scripps Summit Dr, San Diego, CA 92131, United States.
  • Anderson G; Dart Neuroscience, 12278 Scripps Summit Dr, San Diego, CA 92131, United States.
  • Barido R; Dart Neuroscience, 12278 Scripps Summit Dr, San Diego, CA 92131, United States.
  • Basinger J; Dart Neuroscience, 12278 Scripps Summit Dr, San Diego, CA 92131, United States.
  • Bellows CL; Dart Neuroscience, 12278 Scripps Summit Dr, San Diego, CA 92131, United States.
  • Bookser BC; Dart Neuroscience, 12278 Scripps Summit Dr, San Diego, CA 92131, United States.
  • Broadbent NJ; Dart Neuroscience, 12278 Scripps Summit Dr, San Diego, CA 92131, United States.
  • Cabebe C; Dart Neuroscience, 12278 Scripps Summit Dr, San Diego, CA 92131, United States.
  • Chai CK; Dart Neuroscience, 12278 Scripps Summit Dr, San Diego, CA 92131, United States.
  • Chen M; Dart Neuroscience, 12278 Scripps Summit Dr, San Diego, CA 92131, United States.
  • Chow S; Dart Neuroscience, 12278 Scripps Summit Dr, San Diego, CA 92131, United States.
  • Chung M; Dart Neuroscience, 12278 Scripps Summit Dr, San Diego, CA 92131, United States.
  • Heger L; Dart Neuroscience, 12278 Scripps Summit Dr, San Diego, CA 92131, United States.
  • Danks AM; Dart Neuroscience, 12278 Scripps Summit Dr, San Diego, CA 92131, United States.
  • Freestone GC; Dart Neuroscience, 12278 Scripps Summit Dr, San Diego, CA 92131, United States.
  • Gitnick D; Dart Neuroscience, 12278 Scripps Summit Dr, San Diego, CA 92131, United States.
  • Gupta V; Dart Neuroscience, 12278 Scripps Summit Dr, San Diego, CA 92131, United States.
  • Hoffmaster C; Dart Neuroscience, 12278 Scripps Summit Dr, San Diego, CA 92131, United States.
  • Kaplan AP; Dart Neuroscience, 12278 Scripps Summit Dr, San Diego, CA 92131, United States.
  • Kennedy MR; Dart Neuroscience, 12278 Scripps Summit Dr, San Diego, CA 92131, United States.
  • Lee D; Dart Neuroscience, 12278 Scripps Summit Dr, San Diego, CA 92131, United States.
  • Limberis J; Dart Neuroscience, 12278 Scripps Summit Dr, San Diego, CA 92131, United States.
  • Ly K; Dart Neuroscience, 12278 Scripps Summit Dr, San Diego, CA 92131, United States.
  • Mak CC; Dart Neuroscience, 12278 Scripps Summit Dr, San Diego, CA 92131, United States.
  • Masatsugu B; Dart Neuroscience, 12278 Scripps Summit Dr, San Diego, CA 92131, United States.
  • Morse AC; Dart Neuroscience, 12278 Scripps Summit Dr, San Diego, CA 92131, United States.
  • Na J; Dart Neuroscience, 12278 Scripps Summit Dr, San Diego, CA 92131, United States.
  • Neul D; Dart Neuroscience, 12278 Scripps Summit Dr, San Diego, CA 92131, United States.
  • Nikpur J; Dart Neuroscience, 12278 Scripps Summit Dr, San Diego, CA 92131, United States.
  • Renick J; Dart Neuroscience, 12278 Scripps Summit Dr, San Diego, CA 92131, United States.
  • Sebring K; Dart Neuroscience, 12278 Scripps Summit Dr, San Diego, CA 92131, United States.
  • Sevidal S; Dart Neuroscience, 12278 Scripps Summit Dr, San Diego, CA 92131, United States.
  • Tabatabaei A; Dart Neuroscience, 12278 Scripps Summit Dr, San Diego, CA 92131, United States.
  • Wen J; Dart Neuroscience, 12278 Scripps Summit Dr, San Diego, CA 92131, United States.
  • Xia S; Dart Neuroscience, 12278 Scripps Summit Dr, San Diego, CA 92131, United States.
  • Yan Y; Dart Neuroscience, 12278 Scripps Summit Dr, San Diego, CA 92131, United States.
  • Yoder ZW; Dart Neuroscience, 12278 Scripps Summit Dr, San Diego, CA 92131, United States.
  • Zook D; Dart Neuroscience, 12278 Scripps Summit Dr, San Diego, CA 92131, United States.
  • Peters M; Dart Neuroscience, 12278 Scripps Summit Dr, San Diego, CA 92131, United States.
  • Breitenbucher JG; Dart Neuroscience, 12278 Scripps Summit Dr, San Diego, CA 92131, United States.
Bioorg Med Chem Lett ; 30(14): 127214, 2020 07 15.
Article en En | MEDLINE | ID: mdl-32527538

Texto completo: 1 Banco de datos: MEDLINE Asunto principal: Azetidinas / Proteínas de Transporte de Glicina en la Membrana Plasmática / Memoria Límite: Humans Idioma: En Año: 2020 Tipo del documento: Article

Texto completo: 1 Banco de datos: MEDLINE Asunto principal: Azetidinas / Proteínas de Transporte de Glicina en la Membrana Plasmática / Memoria Límite: Humans Idioma: En Año: 2020 Tipo del documento: Article