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Are heterobivalent GRPR- and VPAC1R-bispecific radiopeptides suitable for efficient in vivo tumor imaging of prostate carcinomas?
Lindner, Simon; Rudolf, Henning; Palumbo, Giovanna; Oos, Rosel; Antons, Melissa; Hübner, Ralph; Bartenstein, Peter; Schirrmacher, Ralf; Wängler, Björn; Wängler, Carmen.
  • Lindner S; Department of Nuclear Medicine, University Hospital Munich, Ludwig Maximilians-University Munich, Marchioninistraße 15, 81377 Munich, Germany.
  • Rudolf H; Molecular Imaging and Radiochemistry, Department of Clinical Radiology and Nuclear Medicine, Medical Faculty Mannheim of Heidelberg University, Theodor-Kutzer-Ufer 1-3, 68167 Mannheim, Germany.
  • Palumbo G; Department of Nuclear Medicine, University Hospital Munich, Ludwig Maximilians-University Munich, Marchioninistraße 15, 81377 Munich, Germany.
  • Oos R; Department of Nuclear Medicine, University Hospital Munich, Ludwig Maximilians-University Munich, Marchioninistraße 15, 81377 Munich, Germany.
  • Antons M; Department of Nuclear Medicine, University Hospital Munich, Ludwig Maximilians-University Munich, Marchioninistraße 15, 81377 Munich, Germany.
  • Hübner R; Biomedical Chemistry, Department of Clinical Radiology and Nuclear Medicine, Medical Faculty Mannheim of Heidelberg University, Theodor-Kutzer-Ufer 1-3, 68167 Mannheim, Germany.
  • Bartenstein P; Department of Nuclear Medicine, University Hospital Munich, Ludwig Maximilians-University Munich, Marchioninistraße 15, 81377 Munich, Germany.
  • Schirrmacher R; Department of Oncology, Division of Oncological Imaging, University of Alberta, 11560 University Avenue, Edmonton, AB T6G 1Z2, Canada.
  • Wängler B; Molecular Imaging and Radiochemistry, Department of Clinical Radiology and Nuclear Medicine, Medical Faculty Mannheim of Heidelberg University, Theodor-Kutzer-Ufer 1-3, 68167 Mannheim, Germany.
  • Wängler C; Biomedical Chemistry, Department of Clinical Radiology and Nuclear Medicine, Medical Faculty Mannheim of Heidelberg University, Theodor-Kutzer-Ufer 1-3, 68167 Mannheim, Germany. Electronic address: Carmen.Waengler@medma.uni-heidelberg.de.
Bioorg Med Chem Lett ; 48: 128241, 2021 09 15.
Article en En | MEDLINE | ID: mdl-34217827

Texto completo: 1 Banco de datos: MEDLINE Asunto principal: Péptidos / Neoplasias de la Próstata / Receptores de Bombesina / Receptores de Tipo I del Polipéptido Intestinal Vasoactivo / Tomografía Computarizada por Tomografía de Emisión de Positrones Límite: Humans / Male Idioma: En Año: 2021 Tipo del documento: Article

Texto completo: 1 Banco de datos: MEDLINE Asunto principal: Péptidos / Neoplasias de la Próstata / Receptores de Bombesina / Receptores de Tipo I del Polipéptido Intestinal Vasoactivo / Tomografía Computarizada por Tomografía de Emisión de Positrones Límite: Humans / Male Idioma: En Año: 2021 Tipo del documento: Article