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Development of potent dimeric inhibitors of GAS41 YEATS domain.
Listunov, Dymytrii; Linhares, Brian M; Kim, EunGi; Winkler, Alyssa; Simes, Miranda L; Weaver, Sidney; Cho, Hyo Je; Rizo, Alexandrea; Zolov, Sergey; Keshamouni, Venkateshwar G; Grembecka, Jolanta; Cierpicki, Tomasz.
  • Listunov D; Department of Pathology, University of Michigan, 1150 West Medical Center Dr, MSRB I, Room 4510D, Ann Arbor, MI 48108, USA.
  • Linhares BM; Department of Pathology, University of Michigan, 1150 West Medical Center Dr, MSRB I, Room 4510D, Ann Arbor, MI 48108, USA.
  • Kim E; Department of Pathology, University of Michigan, 1150 West Medical Center Dr, MSRB I, Room 4510D, Ann Arbor, MI 48108, USA.
  • Winkler A; Department of Pathology, University of Michigan, 1150 West Medical Center Dr, MSRB I, Room 4510D, Ann Arbor, MI 48108, USA.
  • Simes ML; Department of Pathology, University of Michigan, 1150 West Medical Center Dr, MSRB I, Room 4510D, Ann Arbor, MI 48108, USA.
  • Weaver S; Department of Pathology, University of Michigan, 1150 West Medical Center Dr, MSRB I, Room 4510D, Ann Arbor, MI 48108, USA.
  • Cho HJ; Department of Pathology, University of Michigan, 1150 West Medical Center Dr, MSRB I, Room 4510D, Ann Arbor, MI 48108, USA.
  • Rizo A; Department of Pathology, University of Michigan, 1150 West Medical Center Dr, MSRB I, Room 4510D, Ann Arbor, MI 48108, USA.
  • Zolov S; Division of Pulmonary and Critical Care Medicine, Department of Internal Medicine, University of Michigan Medical School, 109 Zina Pitcher Place, Ann Arbor, MI 48109-2670, USA.
  • Keshamouni VG; Division of Pulmonary and Critical Care Medicine, Department of Internal Medicine, University of Michigan Medical School, 109 Zina Pitcher Place, Ann Arbor, MI 48109-2670, USA.
  • Grembecka J; Department of Pathology, University of Michigan, 1150 West Medical Center Dr, MSRB I, Room 4510D, Ann Arbor, MI 48108, USA. Electronic address: jolantag@umich.edu.
  • Cierpicki T; Department of Pathology, University of Michigan, 1150 West Medical Center Dr, MSRB I, Room 4510D, Ann Arbor, MI 48108, USA. Electronic address: tomaszc@umich.edu.
Cell Chem Biol ; 28(12): 1716-1727.e6, 2021 12 16.
Article en En | MEDLINE | ID: mdl-34289376

Texto completo: 1 Banco de datos: MEDLINE Asunto principal: Tiofenos / Factores de Transcripción / Carcinoma de Pulmón de Células no Pequeñas / Amidas / Neoplasias Pulmonares / Antineoplásicos Límite: Female / Humans / Male Idioma: En Año: 2021 Tipo del documento: Article

Texto completo: 1 Banco de datos: MEDLINE Asunto principal: Tiofenos / Factores de Transcripción / Carcinoma de Pulmón de Células no Pequeñas / Amidas / Neoplasias Pulmonares / Antineoplásicos Límite: Female / Humans / Male Idioma: En Año: 2021 Tipo del documento: Article