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Discovery of a Potent and Selective Degrader for USP7.
Pei, Yuan; Fu, Jingfeng; Shi, Yunkai; Zhang, Mengmeng; Luo, Guanghao; Luo, Xiaomin; Song, Ning; Mi, Tian; Yang, Yaxi; Li, Jia; Zhou, Yubo; Zhou, Bing.
  • Pei Y; State Key Laboratory of Drug Research, Shanghai Institute of Materia Medica, Chinese Academy of Sciences, 555 Zu Chong Zhi Road, Shanghai, 201203, China.
  • Fu J; University of Chinese Academy of Sciences, 19 Yuquan Road, Beijing, 100049, China.
  • Shi Y; State Key Laboratory of Drug Research, Shanghai Institute of Materia Medica, Chinese Academy of Sciences, 555 Zu Chong Zhi Road, Shanghai, 201203, China.
  • Zhang M; University of Chinese Academy of Sciences, 19 Yuquan Road, Beijing, 100049, China.
  • Luo G; State Key Laboratory of Drug Research, Shanghai Institute of Materia Medica, Chinese Academy of Sciences, 555 Zu Chong Zhi Road, Shanghai, 201203, China.
  • Luo X; School of Pharmaceutical Science and Technology, Hangzhou Institute for Advanced Study, University of Chinese Academy of Sciences, Hangzhou, 310024, China.
  • Song N; State Key Laboratory of Drug Research, Shanghai Institute of Materia Medica, Chinese Academy of Sciences, 555 Zu Chong Zhi Road, Shanghai, 201203, China.
  • Mi T; State Key Laboratory of Drug Research, Shanghai Institute of Materia Medica, Chinese Academy of Sciences, 555 Zu Chong Zhi Road, Shanghai, 201203, China.
  • Yang Y; School of Pharmaceutical Science and Technology, Hangzhou Institute for Advanced Study, University of Chinese Academy of Sciences, Hangzhou, 310024, China.
  • Li J; University of Chinese Academy of Sciences, 19 Yuquan Road, Beijing, 100049, China.
  • Zhou Y; State Key Laboratory of Drug Research, Shanghai Institute of Materia Medica, Chinese Academy of Sciences, 555 Zu Chong Zhi Road, Shanghai, 201203, China.
  • Zhou B; School of Chinese Materia Medica, Nanjing University of Chinese Medicine, Nanjing, 210023, China.
Angew Chem Int Ed Engl ; 61(33): e202204395, 2022 08 15.
Article en En | MEDLINE | ID: mdl-35691827

Texto completo: 1 Banco de datos: MEDLINE Asunto principal: Proteína p53 Supresora de Tumor / Neoplasias Límite: Humans Idioma: En Año: 2022 Tipo del documento: Article

Texto completo: 1 Banco de datos: MEDLINE Asunto principal: Proteína p53 Supresora de Tumor / Neoplasias Límite: Humans Idioma: En Año: 2022 Tipo del documento: Article