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Sonochemical synthesis and biological evaluation of isoquinolin-1(2H)-one/isoindolin-1-one derivatives: Discovery of a positive ago-allosteric modulator (PAAM) of 5HT2CR.
Sandeep Kumar, Jetta; Naimisha, Rapaka; Thirupataiah, B; Sujeevan Reddy, Gangireddy; Bung, Navneet; Roy, Arijit; Bulusu, Gopalakrishnan; Mishra, Ankita; Yadav, Prem N; Misra, Parimal; Pal, Manojit.
  • Sandeep Kumar J; Dr. Reddy's Institute of Life Sciences, University of Hyderabad Campus, Gachibowli, Hyderabad 500 046, India.
  • Naimisha R; Dr. Reddy's Institute of Life Sciences, University of Hyderabad Campus, Gachibowli, Hyderabad 500 046, India.
  • Thirupataiah B; Dr. Reddy's Institute of Life Sciences, University of Hyderabad Campus, Gachibowli, Hyderabad 500 046, India.
  • Sujeevan Reddy G; Dr. Reddy's Institute of Life Sciences, University of Hyderabad Campus, Gachibowli, Hyderabad 500 046, India.
  • Bung N; TCS Research (Life Sciences Division), Tata Consultancy Services Limited, Hyderabad 500081, India.
  • Roy A; TCS Research (Life Sciences Division), Tata Consultancy Services Limited, Hyderabad 500081, India.
  • Bulusu G; Dr. Reddy's Institute of Life Sciences, University of Hyderabad Campus, Gachibowli, Hyderabad 500 046, India; TCS Research (Life Sciences Division), Tata Consultancy Services Limited, Hyderabad 500081, India; Center for Computational Natural Sciences and Bioinformatics, International Institute of In
  • Mishra A; Neuroscience & Ageing Biology, CSIR-Central Drug Research Institute (CSIR-CDRI), Sector 10, Jankipuram Extension, Sitapur Road, Lucknow 226031, India.
  • Yadav PN; Neuroscience & Ageing Biology, CSIR-Central Drug Research Institute (CSIR-CDRI), Sector 10, Jankipuram Extension, Sitapur Road, Lucknow 226031, India.
  • Misra P; Dr. Reddy's Institute of Life Sciences, University of Hyderabad Campus, Gachibowli, Hyderabad 500 046, India. Electronic address: ParimalM@DRILS.ORG.
  • Pal M; Dr. Reddy's Institute of Life Sciences, University of Hyderabad Campus, Gachibowli, Hyderabad 500 046, India. Electronic address: manojitpal@rediffmail.com.
Bioorg Chem ; 129: 106202, 2022 Dec.
Article en En | MEDLINE | ID: mdl-36272252

Texto completo: 1 Banco de datos: MEDLINE Asunto principal: Agonistas del Receptor de Serotonina 5-HT2 / Indoles / Isoquinolinas Tipo de estudio: Prognostic_studies Límite: Animals Idioma: En Año: 2022 Tipo del documento: Article

Texto completo: 1 Banco de datos: MEDLINE Asunto principal: Agonistas del Receptor de Serotonina 5-HT2 / Indoles / Isoquinolinas Tipo de estudio: Prognostic_studies Límite: Animals Idioma: En Año: 2022 Tipo del documento: Article