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Synthesis and Preclinical Evaluation of Small-Molecule Prostate-Specific Membrane Antigen-Targeted Abiraterone Conjugate.
Machulkin, Aleksei E; Nimenko, Ekaterina A; Zyk, Nikolay U; Uspenskaia, Anastasiia A; Smirnova, Galina B; Khan, Irina I; Pokrovsky, Vadim S; Vaneev, Alexander N; Timoshenko, Roman V; Mamed-Nabizade, Vugara V; Zavertkina, Maria V; Erofeev, Alexander; Gorelkin, Petr; Majouga, Alexander G; Zyk, Nikolay V; Khazanova, Elena S; Beloglazkina, Elena K.
  • Machulkin AE; Chemistry Department, Lomonosov Moscow State University, Leninskie Gory, Building 1/3, GSP-1, 119991 Moscow, Russia.
  • Nimenko EA; Chemistry Department, Lomonosov Moscow State University, Leninskie Gory, Building 1/3, GSP-1, 119991 Moscow, Russia.
  • Zyk NU; Chemistry Department, Lomonosov Moscow State University, Leninskie Gory, Building 1/3, GSP-1, 119991 Moscow, Russia.
  • Uspenskaia AA; Chemistry Department, Lomonosov Moscow State University, Leninskie Gory, Building 1/3, GSP-1, 119991 Moscow, Russia.
  • Smirnova GB; N.N. Blokhin Russian Cancer Research Center, 24 Kashirskoye sh., 115478 Moscow, Russia.
  • Khan II; N.N. Blokhin Russian Cancer Research Center, 24 Kashirskoye sh., 115478 Moscow, Russia.
  • Pokrovsky VS; Biochemistry Department, RUDN University, Miklukho-Maklaya Str.6, 117198 Moscow, Russia.
  • Vaneev AN; N.N. Blokhin Russian Cancer Research Center, 24 Kashirskoye sh., 115478 Moscow, Russia.
  • Timoshenko RV; Biochemistry Department, RUDN University, Miklukho-Maklaya Str.6, 117198 Moscow, Russia.
  • Mamed-Nabizade VV; Chemistry Department, Lomonosov Moscow State University, Leninskie Gory, Building 1/3, GSP-1, 119991 Moscow, Russia.
  • Zavertkina MV; Laboratory of Biophysics, National University of Science and Technology MISiS, 4 Leninskiy pr, 119049 Moscow, Russia.
  • Erofeev A; Laboratory of Biophysics, National University of Science and Technology MISiS, 4 Leninskiy pr, 119049 Moscow, Russia.
  • Gorelkin P; Laboratory of Biophysics, National University of Science and Technology MISiS, 4 Leninskiy pr, 119049 Moscow, Russia.
  • Majouga AG; Chemistry Department, Lomonosov Moscow State University, Leninskie Gory, Building 1/3, GSP-1, 119991 Moscow, Russia.
  • Zyk NV; Chemistry Department, Lomonosov Moscow State University, Leninskie Gory, Building 1/3, GSP-1, 119991 Moscow, Russia.
  • Khazanova ES; Laboratory of Biophysics, National University of Science and Technology MISiS, 4 Leninskiy pr, 119049 Moscow, Russia.
  • Beloglazkina EK; Laboratory of Biophysics, National University of Science and Technology MISiS, 4 Leninskiy pr, 119049 Moscow, Russia.
Molecules ; 27(24)2022 Dec 12.
Article en En | MEDLINE | ID: mdl-36557929

Texto completo: 1 Banco de datos: MEDLINE Asunto principal: Neoplasias de la Próstata Límite: Humans / Male Idioma: En Año: 2022 Tipo del documento: Article

Texto completo: 1 Banco de datos: MEDLINE Asunto principal: Neoplasias de la Próstata Límite: Humans / Male Idioma: En Año: 2022 Tipo del documento: Article