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Novel 4-(2-arylidenehydrazineyl)thienopyrimidine derivatives as anticancer EGFR inhibitors: Design, synthesis, biological evaluation, kinome selectivity and in silico insights.
Elsebaie, Heba A; El-Bastawissy, Eman A; Elberembally, Kamel M; Khaleel, Eman F; Badi, Rehab Mustafa; Shaldam, Moataz A; Eldehna, Wagdy M; Tawfik, Haytham O; El-Moselhy, Tarek F.
  • Elsebaie HA; Department of Pharmaceutical Chemistry, Faculty of Pharmacy, Tanta University, Tanta 31527 Egypt. Electronic address: heba.nseer@pharm.tanta.edu.eg.
  • El-Bastawissy EA; Department of Pharmaceutical Chemistry, Faculty of Pharmacy, Tanta University, Tanta 31527 Egypt. Electronic address: emanesmat@pharm.tanta.edu.eg.
  • Elberembally KM; Department of Pharmaceutical Chemistry, Faculty of Pharmacy, Tanta University, Tanta 31527 Egypt. Electronic address: kamel.mohamed@pharm.tanta.edu.eg.
  • Khaleel EF; Department of Medical Physiology, College of Medicine, King Khalid University, King Khalid University, Asir 61421, Saudi Arabia. Electronic address: eman_4000@hotmail.com.
  • Badi RM; Department of Medical Physiology, College of Medicine, King Khalid University, King Khalid University, Asir 61421, Saudi Arabia. Electronic address: rbadi@kku.edu.sa.
  • Shaldam MA; Department of Pharmaceutical Chemistry, Faculty of Pharmacy, Kafrelsheikh University, Kafrelsheikh 33516, Egypt. Electronic address: dr_moutaz_986@pharm.kfs.edu.eg.
  • Eldehna WM; Department of Pharmaceutical Chemistry, Faculty of Pharmacy, Kafrelsheikh University, Kafrelsheikh 33516, Egypt; School of Biotechnology, Badr University in Cairo, Badr City 11829, Egypt. Electronic address: wagdy2000@gmail.com.
  • Tawfik HO; Department of Pharmaceutical Chemistry, Faculty of Pharmacy, Tanta University, Tanta 31527 Egypt. Electronic address: haytham.omar.mahmoud@pharm.tanta.edu.eg.
  • El-Moselhy TF; Department of Pharmaceutical Chemistry, Faculty of Pharmacy, Tanta University, Tanta 31527 Egypt. Electronic address: tarek.faathy@pharm.tanta.edu.eg.
Bioorg Chem ; 140: 106799, 2023 11.
Article en En | MEDLINE | ID: mdl-37625210

Texto completo: 1 Banco de datos: MEDLINE Asunto principal: Apoptosis / Antihipertensivos Idioma: En Año: 2023 Tipo del documento: Article

Texto completo: 1 Banco de datos: MEDLINE Asunto principal: Apoptosis / Antihipertensivos Idioma: En Año: 2023 Tipo del documento: Article