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Discovery and Characterization of ZL-2201, a Potent, Highly Selective, and Orally Bioavailable Small-molecule DNA-PK Inhibitor.
Lal, Shruti; Bhola, Neil E; Sun, Bee-Chun; Chen, Yuping; Huang, Tom; Morton, Vivian; Chen, Kevin X; Xia, Shanghua; Zhang, Haoyu; Parikh, Nehal S; Ye, Qiuping; Veiby, O Petter; Bellovin, David I; Ji, Yuhua.
  • Lal S; Biologics Discovery, Zai Lab (US) LLC, Menlo Park, California.
  • Bhola NE; Biologics Discovery, Zai Lab (US) LLC, Menlo Park, California.
  • Sun BC; Biologics Discovery, Zai Lab (US) LLC, Menlo Park, California.
  • Chen Y; Biologics Discovery, Zai Lab (US) LLC, Menlo Park, California.
  • Huang T; Biologics Discovery, Zai Lab (US) LLC, Menlo Park, California.
  • Morton V; Biologics Discovery, Zai Lab (US) LLC, Menlo Park, California.
  • Chen KX; WuXi AppTec, Shanghai, P.R. China.
  • Xia S; WuXi AppTec, Shanghai, P.R. China.
  • Zhang H; WuXi AppTec, Shanghai, P.R. China.
  • Parikh NS; Biologics Discovery, Zai Lab (US) LLC, Menlo Park, California.
  • Ye Q; Biologics Discovery, Zai Lab (US) LLC, Menlo Park, California.
  • Veiby OP; Biologics Discovery, Zai Lab (US) LLC, Menlo Park, California.
  • Bellovin DI; Biologics Discovery, Zai Lab (US) LLC, Menlo Park, California.
  • Ji Y; Biologics Discovery, Zai Lab (US) LLC, Menlo Park, California.
Cancer Res Commun ; 3(9): 1731-1742, 2023 09.
Article en En | MEDLINE | ID: mdl-37663435

Texto completo: 1 Banco de datos: MEDLINE Asunto principal: Proteína Quinasa Activada por ADN Tipo de estudio: Prognostic_studies Límite: Animals / Humans Idioma: En Año: 2023 Tipo del documento: Article

Texto completo: 1 Banco de datos: MEDLINE Asunto principal: Proteína Quinasa Activada por ADN Tipo de estudio: Prognostic_studies Límite: Animals / Humans Idioma: En Año: 2023 Tipo del documento: Article