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Design and Synthesis of Novel 2-Acetamido, 6-Carboxamide Substituted Benzothiazoles as Potential BRAFV600E Inhibitors - In vitro Evaluation of their Antiproliferative Activity.
Batsi, Yakinthi; Antonopoulou, Georgia; Fotopoulou, Theano; Koumaki, Kassandra; Kritsi, Eftichia; Potamitis, Constantinos; Goulielmaki, Maria; Skarmalioraki, Salomi; Papalouka, Chara; Poulou-Sidiropoulou, Eleni; Kosmidou, Vivian; Douna, Stavroula; Vidali, Maria-Sofia; Gkotsi, Eleni-Fani; Chatziioannou, Aristotelis; Souliotis, Vassilis L; Pletsa, Vasiliki; Papadodima, Olga; Zoumpourlis, Vassilis; Georgiadis, Panagiotis; Zervou, Maria; Pintzas, Alexander; Kostas, Ioannis D.
  • Batsi Y; Institute of Chemical Biology, National Hellenic Research Foundation, Vas. Constantinou Ave. 48, 11635, Athens, Greece.
  • Antonopoulou G; Institute of Chemical Biology, National Hellenic Research Foundation, Vas. Constantinou Ave. 48, 11635, Athens, Greece.
  • Fotopoulou T; Institute of Chemical Biology, National Hellenic Research Foundation, Vas. Constantinou Ave. 48, 11635, Athens, Greece.
  • Koumaki K; Institute of Chemical Biology, National Hellenic Research Foundation, Vas. Constantinou Ave. 48, 11635, Athens, Greece.
  • Kritsi E; Institute of Chemical Biology, National Hellenic Research Foundation, Vas. Constantinou Ave. 48, 11635, Athens, Greece.
  • Potamitis C; Institute of Chemical Biology, National Hellenic Research Foundation, Vas. Constantinou Ave. 48, 11635, Athens, Greece.
  • Goulielmaki M; Institute of Chemical Biology, National Hellenic Research Foundation, Vas. Constantinou Ave. 48, 11635, Athens, Greece.
  • Skarmalioraki S; Institute of Chemical Biology, National Hellenic Research Foundation, Vas. Constantinou Ave. 48, 11635, Athens, Greece.
  • Papalouka C; Institute of Chemical Biology, National Hellenic Research Foundation, Vas. Constantinou Ave. 48, 11635, Athens, Greece.
  • Poulou-Sidiropoulou E; Institute of Chemical Biology, National Hellenic Research Foundation, Vas. Constantinou Ave. 48, 11635, Athens, Greece.
  • Kosmidou V; Institute of Chemical Biology, National Hellenic Research Foundation, Vas. Constantinou Ave. 48, 11635, Athens, Greece.
  • Douna S; Institute of Chemical Biology, National Hellenic Research Foundation, Vas. Constantinou Ave. 48, 11635, Athens, Greece.
  • Vidali MS; Institute of Chemical Biology, National Hellenic Research Foundation, Vas. Constantinou Ave. 48, 11635, Athens, Greece.
  • Gkotsi EF; Institute of Chemical Biology, National Hellenic Research Foundation, Vas. Constantinou Ave. 48, 11635, Athens, Greece.
  • Chatziioannou A; Institute of Chemical Biology, National Hellenic Research Foundation, Vas. Constantinou Ave. 48, 11635, Athens, Greece.
  • Souliotis VL; Institute of Chemical Biology, National Hellenic Research Foundation, Vas. Constantinou Ave. 48, 11635, Athens, Greece.
  • Pletsa V; Institute of Chemical Biology, National Hellenic Research Foundation, Vas. Constantinou Ave. 48, 11635, Athens, Greece.
  • Papadodima O; Institute of Chemical Biology, National Hellenic Research Foundation, Vas. Constantinou Ave. 48, 11635, Athens, Greece.
  • Zoumpourlis V; Institute of Chemical Biology, National Hellenic Research Foundation, Vas. Constantinou Ave. 48, 11635, Athens, Greece.
  • Georgiadis P; Institute of Chemical Biology, National Hellenic Research Foundation, Vas. Constantinou Ave. 48, 11635, Athens, Greece.
  • Zervou M; Institute of Chemical Biology, National Hellenic Research Foundation, Vas. Constantinou Ave. 48, 11635, Athens, Greece.
  • Pintzas A; Institute of Chemical Biology, National Hellenic Research Foundation, Vas. Constantinou Ave. 48, 11635, Athens, Greece.
  • Kostas ID; Institute of Chemical Biology, National Hellenic Research Foundation, Vas. Constantinou Ave. 48, 11635, Athens, Greece.
ChemMedChem ; 18(22): e202300322, 2023 11 16.
Article en En | MEDLINE | ID: mdl-37792577

Texto completo: 1 Banco de datos: MEDLINE Asunto principal: Benzotiazoles / Antineoplásicos Idioma: En Año: 2023 Tipo del documento: Article

Texto completo: 1 Banco de datos: MEDLINE Asunto principal: Benzotiazoles / Antineoplásicos Idioma: En Año: 2023 Tipo del documento: Article