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Rational Screening for Cooperativity in Small-Molecule Inducers of Protein-Protein Associations.
Liu, Shuang; Tong, Bingqi; Mason, Jeremy W; Ostrem, Jonathan M; Tutter, Antonin; Hua, Bruce K; Tang, Sunny A; Bonazzi, Simone; Briner, Karin; Berst, Frédéric; Zécri, Frédéric J; Schreiber, Stuart L.
  • Liu S; Chemical Biology and Therapeutics Science, Broad Institute of MIT and Harvard, 415 Main Street, Cambridge, Massachusetts 02142, United States.
  • Tong B; Department of Chemistry and Chemical Biology, Harvard University, 12 Oxford Street, Cambridge, Massachusetts 02138, United States.
  • Mason JW; Chemical Biology and Therapeutics Science, Broad Institute of MIT and Harvard, 415 Main Street, Cambridge, Massachusetts 02142, United States.
  • Ostrem JM; Department of Chemistry and Chemical Biology, Harvard University, 12 Oxford Street, Cambridge, Massachusetts 02138, United States.
  • Tutter A; Global Discovery Chemistry, Novartis Institutes for BioMedical Research, 181 Massachusetts Avenue, Cambridge, Massachusetts 02139, United States.
  • Hua BK; Chemical Biology and Therapeutics Science, Broad Institute of MIT and Harvard, 415 Main Street, Cambridge, Massachusetts 02142, United States.
  • Tang SA; Global Discovery Chemistry, Novartis Institutes for BioMedical Research, 181 Massachusetts Avenue, Cambridge, Massachusetts 02139, United States.
  • Bonazzi S; Chemical Biology and Therapeutics Science, Broad Institute of MIT and Harvard, 415 Main Street, Cambridge, Massachusetts 02142, United States.
  • Briner K; Chemical Biology and Therapeutics, Novartis Institutes for BioMedical Research, 181 Massachusetts Avenue, Cambridge, Massachusetts 02139, United States.
  • Berst F; Chemical Biology and Therapeutics Science, Broad Institute of MIT and Harvard, 415 Main Street, Cambridge, Massachusetts 02142, United States.
  • Zécri FJ; Department of Chemistry and Chemical Biology, Harvard University, 12 Oxford Street, Cambridge, Massachusetts 02138, United States.
  • Schreiber SL; Department of Chemistry and Chemical Biology, Harvard University, 12 Oxford Street, Cambridge, Massachusetts 02138, United States.
J Am Chem Soc ; 145(42): 23281-23291, 2023 10 25.
Article en En | MEDLINE | ID: mdl-37816014

Texto completo: 1 Banco de datos: MEDLINE Asunto principal: ADN / Proteínas Tipo de estudio: Diagnostic_studies / Risk_factors_studies / Screening_studies Idioma: En Año: 2023 Tipo del documento: Article

Texto completo: 1 Banco de datos: MEDLINE Asunto principal: ADN / Proteínas Tipo de estudio: Diagnostic_studies / Risk_factors_studies / Screening_studies Idioma: En Año: 2023 Tipo del documento: Article