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A novel N-heterocycles substituted oseltamivir derivatives as potent inhibitors of influenza virus neuraminidase: discovery, synthesis and biological evaluation.
Zhang, Jiwei; Liu, Chuanfeng; Jia, Ruifang; Zhang, Xujie; Zhang, Jian; Bertagnin, Chiara; Bonomini, Anna; Guizzo, Laura; Jiang, Yuanmin; Jia, Huinan; Jia, Shuzhen; Ma, Xiuli; Loregian, Arianna; Huang, Bing; Zhan, Peng; Liu, Xinyong.
  • Zhang J; Department of Medicinal Chemistry, Key Laboratory of Chemical Biology (Ministry of Education), School of Pharmaceutical Sciences, Cheeloo College of Medicine, Shandong University, Jinan, Shandong, P.R. China.
  • Liu C; Department of Medicinal Chemistry, Key Laboratory of Chemical Biology (Ministry of Education), School of Pharmaceutical Sciences, Cheeloo College of Medicine, Shandong University, Jinan, Shandong, P.R. China.
  • Jia R; Suzhou Research Institute of Shandong University, Suzhou, Jiangsu, P.R. China.
  • Zhang X; Department of Medicinal Chemistry, Key Laboratory of Chemical Biology (Ministry of Education), School of Pharmaceutical Sciences, Cheeloo College of Medicine, Shandong University, Jinan, Shandong, P.R. China.
  • Zhang J; Department of Medicinal Chemistry, Key Laboratory of Chemical Biology (Ministry of Education), School of Pharmaceutical Sciences, Cheeloo College of Medicine, Shandong University, Jinan, Shandong, P.R. China.
  • Bertagnin C; Institute of Medical Sciences, The Second Hospital, Shandong University, Jinan, Shandong, P.R. China.
  • Bonomini A; Department of Molecular Medicine, University of Padova, Padova, Italy.
  • Guizzo L; Department of Molecular Medicine, University of Padova, Padova, Italy.
  • Jiang Y; Department of Molecular Medicine, University of Padova, Padova, Italy.
  • Jia H; Department of Medicinal Chemistry, Key Laboratory of Chemical Biology (Ministry of Education), School of Pharmaceutical Sciences, Cheeloo College of Medicine, Shandong University, Jinan, Shandong, P.R. China.
  • Jia S; Department of Medicinal Chemistry, Key Laboratory of Chemical Biology (Ministry of Education), School of Pharmaceutical Sciences, Cheeloo College of Medicine, Shandong University, Jinan, Shandong, P.R. China.
  • Ma X; Department of Medicinal Chemistry, Key Laboratory of Chemical Biology (Ministry of Education), School of Pharmaceutical Sciences, Cheeloo College of Medicine, Shandong University, Jinan, Shandong, P.R. China.
  • Loregian A; Institute of Poultry Science, Shandong Academy of Agricultural Sciences, Jinan, Shandong, P.R. China.
  • Huang B; Department of Molecular Medicine, University of Padova, Padova, Italy.
  • Zhan P; Institute of Poultry Science, Shandong Academy of Agricultural Sciences, Jinan, Shandong, P.R. China.
  • Liu X; Department of Medicinal Chemistry, Key Laboratory of Chemical Biology (Ministry of Education), School of Pharmaceutical Sciences, Cheeloo College of Medicine, Shandong University, Jinan, Shandong, P.R. China.
J Enzyme Inhib Med Chem ; 38(1): 2277135, 2023 Dec.
Article en En | MEDLINE | ID: mdl-37955306

Texto completo: 1 Banco de datos: MEDLINE Asunto principal: Subtipo H1N1 del Virus de la Influenza A / Subtipo H5N1 del Virus de la Influenza A Idioma: En Año: 2023 Tipo del documento: Article

Texto completo: 1 Banco de datos: MEDLINE Asunto principal: Subtipo H1N1 del Virus de la Influenza A / Subtipo H5N1 del Virus de la Influenza A Idioma: En Año: 2023 Tipo del documento: Article