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A recombinant approach for stapled peptide discovery yields inhibitors of the RAD51 recombinase.
Pantelejevs, Teodors; Zuazua-Villar, Pedro; Koczy, Oliwia; Counsell, Andrew J; Walsh, Stephen J; Robertson, Naomi S; Spring, David R; Downs, Jessica A; Hyvönen, Marko.
  • Pantelejevs T; Department of Biochemistry, University of Cambridge CB2 1GA UK teodors.pantelejevs@osi.lv mh256@cam.ac.uk.
  • Zuazua-Villar P; Latvian Institute of Organic Synthesis Aizkraukles 21 Riga LV-1006 Latvia.
  • Koczy O; Division of Cancer Biology, The Institute of Cancer Research London SW3 6JB UK.
  • Counsell AJ; Department of Biochemistry, University of Cambridge CB2 1GA UK teodors.pantelejevs@osi.lv mh256@cam.ac.uk.
  • Walsh SJ; Yusuf Hamied Department of Chemistry, University of Cambridge CB2 1EW UK.
  • Robertson NS; Yusuf Hamied Department of Chemistry, University of Cambridge CB2 1EW UK.
  • Spring DR; Yusuf Hamied Department of Chemistry, University of Cambridge CB2 1EW UK.
  • Downs JA; Yusuf Hamied Department of Chemistry, University of Cambridge CB2 1EW UK.
  • Hyvönen M; Division of Cancer Biology, The Institute of Cancer Research London SW3 6JB UK.
Chem Sci ; 14(47): 13915-13923, 2023 Dec 06.
Article en En | MEDLINE | ID: mdl-38075664