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Discovery of Novel Putative Inhibitors of UDP-GlcNAc 2-Epimerase as Potent Antibacterial Agents.
Xu, Yong; Brenning, Benjamin; Clifford, Adrianne; Vollmer, David; Bearss, Jared; Jones, Carissa; McCarthy, Virgil; Shi, Chongtie; Wolfe, Bradley; Aavula, Bhasker; Warner, Steve; Bearss, David J; McCullar, Michael V; Schuch, Raymond; Pelzek, Adam; Bhaskaran, Shyam S; Stebbins, C Erec; Goldberg, Allan R; Fischetti, Vincent A; Vankayalapati, Hariprasad.
Afiliação
  • Xu Y; Astex Pharmaceuticals, Inc. (formerly known as SuperGen, Inc.), 4140 Dublin Boulevard, Suite 200, Dublin, CA 94568, U.S.A.
  • Brenning B; Astex Pharmaceuticals, Inc. (formerly known as SuperGen, Inc.), 4140 Dublin Boulevard, Suite 200, Dublin, CA 94568, U.S.A.
  • Clifford A; Astex Pharmaceuticals, Inc. (formerly known as SuperGen, Inc.), 4140 Dublin Boulevard, Suite 200, Dublin, CA 94568, U.S.A.
  • Vollmer D; Astex Pharmaceuticals, Inc. (formerly known as SuperGen, Inc.), 4140 Dublin Boulevard, Suite 200, Dublin, CA 94568, U.S.A.
  • Bearss J; Astex Pharmaceuticals, Inc. (formerly known as SuperGen, Inc.), 4140 Dublin Boulevard, Suite 200, Dublin, CA 94568, U.S.A ; Division of Oncology of School of Medicine and Center for Investigational Therapeutics at Huntsman Cancer Institute, University of Utah, 2000 Circle of Hope, Salt Lake City, UT
  • Jones C; Astex Pharmaceuticals, Inc. (formerly known as SuperGen, Inc.), 4140 Dublin Boulevard, Suite 200, Dublin, CA 94568, U.S.A.
  • McCarthy V; Astex Pharmaceuticals, Inc. (formerly known as SuperGen, Inc.), 4140 Dublin Boulevard, Suite 200, Dublin, CA 94568, U.S.A.
  • Shi C; Astex Pharmaceuticals, Inc. (formerly known as SuperGen, Inc.), 4140 Dublin Boulevard, Suite 200, Dublin, CA 94568, U.S.A.
  • Wolfe B; Astex Pharmaceuticals, Inc. (formerly known as SuperGen, Inc.), 4140 Dublin Boulevard, Suite 200, Dublin, CA 94568, U.S.A.
  • Aavula B; Astex Pharmaceuticals, Inc. (formerly known as SuperGen, Inc.), 4140 Dublin Boulevard, Suite 200, Dublin, CA 94568, U.S.A.
  • Warner S; Astex Pharmaceuticals, Inc. (formerly known as SuperGen, Inc.), 4140 Dublin Boulevard, Suite 200, Dublin, CA 94568, U.S.A.
  • Bearss DJ; Astex Pharmaceuticals, Inc. (formerly known as SuperGen, Inc.), 4140 Dublin Boulevard, Suite 200, Dublin, CA 94568, U.S.A ; Division of Oncology of School of Medicine and Center for Investigational Therapeutics at Huntsman Cancer Institute, University of Utah, 2000 Circle of Hope, Salt Lake City, UT
  • McCullar MV; Astex Pharmaceuticals, Inc. (formerly known as SuperGen, Inc.), 4140 Dublin Boulevard, Suite 200, Dublin, CA 94568, U.S.A.
  • Schuch R; Laboratory of Bacterial Pathogenesis and Immunology, The Rockefeller University, New York, NY 10065, U.S.A.
  • Pelzek A; Laboratory of Bacterial Pathogenesis and Immunology, The Rockefeller University, New York, NY 10065, U.S.A.
  • Bhaskaran SS; Laboratory of Bacterial Pathogenesis and Immunology, The Rockefeller University, New York, NY 10065, U.S.A.
  • Stebbins CE; Laboratory of Structural Microbiology, The Rockefeller University, New York, NY, U.S.A.
  • Goldberg AR; Astex Pharmaceuticals, Inc. (formerly known as SuperGen, Inc.), 4140 Dublin Boulevard, Suite 200, Dublin, CA 94568, U.S.A ; Avacyn Pharmaceuticals, Inc., Teaneck, NJ, U.S.A. (Current Address).
  • Fischetti VA; Laboratory of Bacterial Pathogenesis and Immunology, The Rockefeller University, New York, NY 10065, U.S.A.
  • Vankayalapati H; Astex Pharmaceuticals, Inc. (formerly known as SuperGen, Inc.), 4140 Dublin Boulevard, Suite 200, Dublin, CA 94568, U.S.A ; Division of Oncology of School of Medicine and Center for Investigational Therapeutics at Huntsman Cancer Institute, University of Utah, 2000 Circle of Hope, Salt Lake City, UT
ACS Med Chem Lett ; 4(12): 1142-1147, 2013 Dec 12.
Article em En | MEDLINE | ID: mdl-24443700

Texto completo: 1 Base de dados: MEDLINE Idioma: En Ano de publicação: 2013 Tipo de documento: Article

Texto completo: 1 Base de dados: MEDLINE Idioma: En Ano de publicação: 2013 Tipo de documento: Article