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Endomorphin analogues with mixed µ-opioid (MOP) receptor agonism/δ-opioid (DOP) receptor antagonism and lacking ß-arrestin2 recruitment activity.
Cai, Jun; Song, Bowen; Cai, Yunxin; Ma, Yu; Lam, Ai-Leen; Magiera, Julia; Sekar, Sunder; Wyse, Bruce D; Ambo, Akihiro; Sasaki, Yusuke; Lazarus, Lawrence H; Smith, Maree T; Li, Tingyou.
Afiliação
  • Cai J; School of Pharmacy, Nanjing Medical University, Nanjing 211166, China.
  • Song B; School of Pharmacy, Nanjing Medical University, Nanjing 211166, China.
  • Cai Y; School of Pharmacy, Nanjing Medical University, Nanjing 211166, China.
  • Ma Y; School of Pharmacy, Nanjing Medical University, Nanjing 211166, China.
  • Lam AL; Centre for Integrated Preclinical Drug Development, The University of Queensland, Brisbane, QLD 4072, Australia.
  • Magiera J; Centre for Integrated Preclinical Drug Development, The University of Queensland, Brisbane, QLD 4072, Australia.
  • Sekar S; Centre for Integrated Preclinical Drug Development, The University of Queensland, Brisbane, QLD 4072, Australia.
  • Wyse BD; Centre for Integrated Preclinical Drug Development, The University of Queensland, Brisbane, QLD 4072, Australia.
  • Ambo A; Tohoku Pharmaceutical University, 4-1 Komatsushima 4-chome, Aoba-ku, Sendai 981-8558, Japan.
  • Sasaki Y; Tohoku Pharmaceutical University, 4-1 Komatsushima 4-chome, Aoba-ku, Sendai 981-8558, Japan.
  • Lazarus LH; Medicinal Chemistry Group, Laboratory of Pharmacology and Chemistry, National Institute of Environmental Health Science, Research Triangle Park, NC 27709, USA.
  • Smith MT; Centre for Integrated Preclinical Drug Development, The University of Queensland, Brisbane, QLD 4072, Australia. Electronic address: maree.smith@uq.edu.au.
  • Li T; School of Pharmacy, Nanjing Medical University, Nanjing 211166, China; Collaborative Innovation Center for Cardiovascular Disease Translational Medicine, Nanjing Medical University, Nanjing 211166, China. Electronic address: l_tingyou@njmu.edu.cn.
Bioorg Med Chem ; 22(7): 2208-19, 2014 Apr 01.
Article em En | MEDLINE | ID: mdl-24613457

Texto completo: 1 Base de dados: MEDLINE Assunto principal: Oligopeptídeos / Receptores Opioides delta / Receptores Opioides mu / Arrestinas Limite: Animals / Humans / Male Idioma: En Ano de publicação: 2014 Tipo de documento: Article

Texto completo: 1 Base de dados: MEDLINE Assunto principal: Oligopeptídeos / Receptores Opioides delta / Receptores Opioides mu / Arrestinas Limite: Animals / Humans / Male Idioma: En Ano de publicação: 2014 Tipo de documento: Article