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Discovery of substituted benzamides as follicle stimulating hormone receptor allosteric modulators.
Yu, Henry N; Richardson, Thomas E; Nataraja, Selva; Fischer, David J; Sriraman, Venkataraman; Jiang, Xuliang; Bharathi, Pandi; Foglesong, Robert J; Haxell, Thomas F N; Heasley, Brian H; Jenks, Mathew; Li, Jane; Dugas, Melanie S; Collis, Regina; Tian, Hui; Palmer, Stephen; Goutopoulos, Andreas.
Afiliação
  • Yu HN; EMD Serono Research Institute, 45A Middlesex Turnpike, Billerica, MA 01821, United States; TocopheRx, Inc., Suite 1077, 15 New England Executive Park, Burlington, MA 01803, United States. Electronic address: henry.yu@emdserono.com.
  • Richardson TE; Scynexis, Inc., 3501 C Tricenter Boulevard, Durham, NC 27713, United States.
  • Nataraja S; TocopheRx, Inc., Suite 1077, 15 New England Executive Park, Burlington, MA 01803, United States.
  • Fischer DJ; EMD Serono Research Institute, 45A Middlesex Turnpike, Billerica, MA 01821, United States.
  • Sriraman V; EMD Serono Research Institute, 45A Middlesex Turnpike, Billerica, MA 01821, United States.
  • Jiang X; EMD Serono Research Institute, 45A Middlesex Turnpike, Billerica, MA 01821, United States.
  • Bharathi P; Scynexis, Inc., 3501 C Tricenter Boulevard, Durham, NC 27713, United States.
  • Foglesong RJ; Scynexis, Inc., 3501 C Tricenter Boulevard, Durham, NC 27713, United States.
  • Haxell TF; Scynexis, Inc., 3501 C Tricenter Boulevard, Durham, NC 27713, United States.
  • Heasley BH; Scynexis, Inc., 3501 C Tricenter Boulevard, Durham, NC 27713, United States.
  • Jenks M; Scynexis, Inc., 3501 C Tricenter Boulevard, Durham, NC 27713, United States.
  • Li J; EMD Serono Research Institute, 45A Middlesex Turnpike, Billerica, MA 01821, United States.
  • Dugas MS; EMD Serono Research Institute, 45A Middlesex Turnpike, Billerica, MA 01821, United States.
  • Collis R; EMD Serono Research Institute, 45A Middlesex Turnpike, Billerica, MA 01821, United States.
  • Tian H; EMD Serono Research Institute, 45A Middlesex Turnpike, Billerica, MA 01821, United States.
  • Palmer S; TocopheRx, Inc., Suite 1077, 15 New England Executive Park, Burlington, MA 01803, United States.
  • Goutopoulos A; EMD Serono Research Institute, 45A Middlesex Turnpike, Billerica, MA 01821, United States.
Bioorg Med Chem Lett ; 24(9): 2168-72, 2014 May 01.
Article em En | MEDLINE | ID: mdl-24685543

Texto completo: 1 Base de dados: MEDLINE Assunto principal: Benzamidas / Regulação Alostérica / Hormônio Foliculoestimulante Tipo de estudo: Guideline Limite: Animals / Female / Humans Idioma: En Ano de publicação: 2014 Tipo de documento: Article

Texto completo: 1 Base de dados: MEDLINE Assunto principal: Benzamidas / Regulação Alostérica / Hormônio Foliculoestimulante Tipo de estudo: Guideline Limite: Animals / Female / Humans Idioma: En Ano de publicação: 2014 Tipo de documento: Article