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A new class of multimerization selective inhibitors of HIV-1 integrase.
Sharma, Amit; Slaughter, Alison; Jena, Nivedita; Feng, Lei; Kessl, Jacques J; Fadel, Hind J; Malani, Nirav; Male, Frances; Wu, Li; Poeschla, Eric; Bushman, Frederic D; Fuchs, James R; Kvaratskhelia, Mamuka.
Afiliação
  • Sharma A; Center for Retrovirus Research and College of Pharmacy, The Ohio State University, Columbus, Ohio, United States of America.
  • Slaughter A; Center for Retrovirus Research and College of Pharmacy, The Ohio State University, Columbus, Ohio, United States of America.
  • Jena N; Division of Medicinal Chemistry and Pharmacognosy, College of Pharmacy, The Ohio State University, Columbus, Ohio, United States of America.
  • Feng L; Center for Retrovirus Research and College of Pharmacy, The Ohio State University, Columbus, Ohio, United States of America.
  • Kessl JJ; Center for Retrovirus Research and College of Pharmacy, The Ohio State University, Columbus, Ohio, United States of America.
  • Fadel HJ; Department of Molecular Medicine & Division of Infectious Diseases, Mayo Clinic College of Medicine, Rochester, Minnesota, United States of America.
  • Malani N; Perelman School of Medicine, Department of Microbiology, University of Pennsylvania, Philadelphia, Pennsylvania, United States of America.
  • Male F; Perelman School of Medicine, Department of Microbiology, University of Pennsylvania, Philadelphia, Pennsylvania, United States of America.
  • Wu L; Center for Retrovirus Research and Department of Veterinary Biosciences, The Ohio State University, Columbus, Ohio, United States of America.
  • Poeschla E; Department of Molecular Medicine & Division of Infectious Diseases, Mayo Clinic College of Medicine, Rochester, Minnesota, United States of America.
  • Bushman FD; Perelman School of Medicine, Department of Microbiology, University of Pennsylvania, Philadelphia, Pennsylvania, United States of America.
  • Fuchs JR; Division of Medicinal Chemistry and Pharmacognosy, College of Pharmacy, The Ohio State University, Columbus, Ohio, United States of America.
  • Kvaratskhelia M; Center for Retrovirus Research and College of Pharmacy, The Ohio State University, Columbus, Ohio, United States of America.
PLoS Pathog ; 10(5): e1004171, 2014 May.
Article em En | MEDLINE | ID: mdl-24874515

Texto completo: 1 Base de dados: MEDLINE Assunto principal: Antivirais / Integração Viral / Inibidores de Integrase de HIV / Integrase de HIV / Peptídeos e Proteínas de Sinalização Intercelular / Multimerização Proteica Limite: Humans Idioma: En Ano de publicação: 2014 Tipo de documento: Article

Texto completo: 1 Base de dados: MEDLINE Assunto principal: Antivirais / Integração Viral / Inibidores de Integrase de HIV / Integrase de HIV / Peptídeos e Proteínas de Sinalização Intercelular / Multimerização Proteica Limite: Humans Idioma: En Ano de publicação: 2014 Tipo de documento: Article