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2-Alkyl/alkenyl substituted pyridine C-region analogues of 2-(3-fluoro-4-methylsulfonylaminophenyl)propanamides as highly potent TRPV1 antagonists.
Ryu, HyungChul; Seo, Sejin; Cho, Seong-Hee; Kim, Ho Shin; Jung, Aeran; Kang, Dong Wook; Son, Karam; Cui, Minghua; Hong, Sun-hye; Sharma, Pankaz Kumar; Choi, Sun; Blumberg, Peter M; Frank-Foltyn, Robert; Bahrenberg, Gregor; Stockhausen, Hannelore; Schiene, Klaus; Christoph, Thomas; Frormann, Sven; Lee, Jeewoo.
Afiliação
  • Ryu H; Laboratory of Medicinal Chemistry, Research Institute of Pharmaceutical Sciences, College of Pharmacy, Seoul National University, Seoul 151-742, Republic of Korea.
  • Seo S; Laboratory of Medicinal Chemistry, Research Institute of Pharmaceutical Sciences, College of Pharmacy, Seoul National University, Seoul 151-742, Republic of Korea.
  • Cho SH; Laboratory of Medicinal Chemistry, Research Institute of Pharmaceutical Sciences, College of Pharmacy, Seoul National University, Seoul 151-742, Republic of Korea.
  • Kim HS; Laboratory of Medicinal Chemistry, Research Institute of Pharmaceutical Sciences, College of Pharmacy, Seoul National University, Seoul 151-742, Republic of Korea.
  • Jung A; Laboratory of Medicinal Chemistry, Research Institute of Pharmaceutical Sciences, College of Pharmacy, Seoul National University, Seoul 151-742, Republic of Korea.
  • Kang DW; Laboratory of Medicinal Chemistry, Research Institute of Pharmaceutical Sciences, College of Pharmacy, Seoul National University, Seoul 151-742, Republic of Korea; Department of Pharmaceutical Science and Technology, College of Health and Medical Science, Catholic University of Deagu, Gyeongsan-si,
  • Son K; National Leading Research Lab of Molecular Modeling & Drug Design, College of Pharmacy, Graduate School of Pharmaceutical Sciences, and Global Top 5 Research Program, Ewha Womans University, Seoul 120-750, Republic of Korea.
  • Cui M; National Leading Research Lab of Molecular Modeling & Drug Design, College of Pharmacy, Graduate School of Pharmaceutical Sciences, and Global Top 5 Research Program, Ewha Womans University, Seoul 120-750, Republic of Korea.
  • Hong SH; National Leading Research Lab of Molecular Modeling & Drug Design, College of Pharmacy, Graduate School of Pharmaceutical Sciences, and Global Top 5 Research Program, Ewha Womans University, Seoul 120-750, Republic of Korea.
  • Sharma PK; National Leading Research Lab of Molecular Modeling & Drug Design, College of Pharmacy, Graduate School of Pharmaceutical Sciences, and Global Top 5 Research Program, Ewha Womans University, Seoul 120-750, Republic of Korea.
  • Choi S; National Leading Research Lab of Molecular Modeling & Drug Design, College of Pharmacy, Graduate School of Pharmaceutical Sciences, and Global Top 5 Research Program, Ewha Womans University, Seoul 120-750, Republic of Korea.
  • Blumberg PM; Laboratory of Cancer Biology and Genetics, Center for Cancer Research, National Cancer Institute, NIH, Bethesda, MD 20892, USA.
  • Frank-Foltyn R; Grunenthal Innovation, Grunenthal GmbH, D-52078 Aachen, Germany.
  • Bahrenberg G; Grunenthal Innovation, Grunenthal GmbH, D-52078 Aachen, Germany.
  • Stockhausen H; Grunenthal Innovation, Grunenthal GmbH, D-52078 Aachen, Germany.
  • Schiene K; Grunenthal Innovation, Grunenthal GmbH, D-52078 Aachen, Germany.
  • Christoph T; Grunenthal Innovation, Grunenthal GmbH, D-52078 Aachen, Germany.
  • Frormann S; Grunenthal Innovation, Grunenthal GmbH, D-52078 Aachen, Germany.
  • Lee J; Laboratory of Medicinal Chemistry, Research Institute of Pharmaceutical Sciences, College of Pharmacy, Seoul National University, Seoul 151-742, Republic of Korea. Electronic address: jeewoo@snu.ac.kr.
Bioorg Med Chem Lett ; 24(16): 4039-43, 2014 Aug 15.
Article em En | MEDLINE | ID: mdl-24948568
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Texto completo: 1 Base de dados: MEDLINE Assunto principal: Fenilpropionatos / Piridinas / Canais de Cátion TRPV / Hidrocarbonetos Fluorados Limite: Humans Idioma: En Ano de publicação: 2014 Tipo de documento: Article
Texto completo
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Texto completo: 1 Base de dados: MEDLINE Assunto principal: Fenilpropionatos / Piridinas / Canais de Cátion TRPV / Hidrocarbonetos Fluorados Limite: Humans Idioma: En Ano de publicação: 2014 Tipo de documento: Article