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Expanding the results of a high throughput screen against an isochorismate-pyruvate lyase to enzymes of a similar scaffold or mechanism.
Meneely, Kathleen M; Luo, Qianyi; Riley, Andrew P; Taylor, Byron; Roy, Anuradha; Stein, Ross L; Prisinzano, Thomas E; Lamb, Audrey L.
Afiliação
  • Meneely KM; Department of Molecular Biosciences, University of Kansas, 1200 Sunnyside Ave, Lawrence, KS 66045, United States.
  • Luo Q; Department of Molecular Biosciences, University of Kansas, 1200 Sunnyside Ave, Lawrence, KS 66045, United States.
  • Riley AP; Department of Chemistry, University of Kansas, 1251 Wescoe Hall Dr, Lawrence, KS 66045, United States.
  • Taylor B; High Throughput Screening Facility, University of Kansas, 2034 Becker Dr, Lawrence, KS 66047, United States.
  • Roy A; High Throughput Screening Facility, University of Kansas, 2034 Becker Dr, Lawrence, KS 66047, United States.
  • Stein RL; High Throughput Screening Facility, University of Kansas, 2034 Becker Dr, Lawrence, KS 66047, United States.
  • Prisinzano TE; Department of Medicinal Chemistry, University of Kansas, 1251 Wescoe Hall Dr, Lawrence, KS 66045, United States.
  • Lamb AL; Department of Molecular Biosciences, University of Kansas, 1200 Sunnyside Ave, Lawrence, KS 66045, United States. Electronic address: lamb@ku.edu.
Bioorg Med Chem ; 22(21): 5961-9, 2014 Nov 01.
Article em En | MEDLINE | ID: mdl-25282647

Texto completo: 1 Base de dados: MEDLINE Assunto principal: Pseudomonas aeruginosa / Ácido Corísmico / Inibidores Enzimáticos / Oxo-Ácido-Liases / Antibacterianos Limite: Humans Idioma: En Ano de publicação: 2014 Tipo de documento: Article

Texto completo: 1 Base de dados: MEDLINE Assunto principal: Pseudomonas aeruginosa / Ácido Corísmico / Inibidores Enzimáticos / Oxo-Ácido-Liases / Antibacterianos Limite: Humans Idioma: En Ano de publicação: 2014 Tipo de documento: Article