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A new crystal structure fragment-based pharmacophore method for G protein-coupled receptors.
Fidom, Kimberley; Isberg, Vignir; Hauser, Alexander S; Mordalski, Stefan; Lehto, Thomas; Bojarski, Andrzej J; Gloriam, David E.
Afiliação
  • Fidom K; Department of Drug Design and Pharmacology, Faculty of Health and Medical Sciences, University of Copenhagen, Denmark. Electronic address: kimberleyfidom@gmail.com.
  • Isberg V; Department of Drug Design and Pharmacology, Faculty of Health and Medical Sciences, University of Copenhagen, Denmark. Electronic address: vis@sund.ku.dk.
  • Hauser AS; Department of Drug Design and Pharmacology, Faculty of Health and Medical Sciences, University of Copenhagen, Denmark. Electronic address: alexshauser@gmail.com.
  • Mordalski S; Department of Medicinal Chemistry, Institute of Pharmacology, Polish Academy of Sciences, Poland; Faculty of Biochemistry, Biophysics and Biotechnology, Jagiellonian University, Krakow, Poland. Electronic address: stefanm@if-pan.krakow.pl.
  • Lehto T; Department of Drug Design and Pharmacology, Faculty of Health and Medical Sciences, University of Copenhagen, Denmark. Electronic address: thomas@leh2.dk.
  • Bojarski AJ; Department of Medicinal Chemistry, Institute of Pharmacology, Polish Academy of Sciences, Poland. Electronic address: bojarski@if-pan.krakow.pl.
  • Gloriam DE; Department of Drug Design and Pharmacology, Faculty of Health and Medical Sciences, University of Copenhagen, Denmark. Electronic address: david.gloriam@sund.ku.dk.
Methods ; 71: 104-12, 2015 Jan.
Article em En | MEDLINE | ID: mdl-25286328

Texto completo: 1 Base de dados: MEDLINE Assunto principal: Modelos Moleculares / Cristalografia por Raios X / Receptores Acoplados a Proteínas G Idioma: En Ano de publicação: 2015 Tipo de documento: Article

Texto completo: 1 Base de dados: MEDLINE Assunto principal: Modelos Moleculares / Cristalografia por Raios X / Receptores Acoplados a Proteínas G Idioma: En Ano de publicação: 2015 Tipo de documento: Article