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Molecular docking study, synthesis and biological evaluation of Mannich bases as Hsp90 inhibitors.
Dutta Gupta, Sayan; Bommaka, Manish Kumar; Mazaira, Gisela I; Galigniana, Mario D; Subrahmanyam, Chavali Venkata Satya; Gowrishankar, Naryanasamy Lachmana; Raghavendra, Nulgumnalli Manjunathaiah.
Afiliação
  • Dutta Gupta S; Department of Pharmaceutical Chemistry, Gokaraju Rangaraju College of Pharmacy, Osmania University, Hyderabad, India; R&D Centre, Department of Pharmaceutical Sciences, Jawaharlal Nehru Technological University, Hyderabad, India.
  • Bommaka MK; Department of Pharmaceutical Chemistry, Gokaraju Rangaraju College of Pharmacy, Osmania University, Hyderabad, India.
  • Mazaira GI; Department of Biological Chemistry, Faculty of Natural Sciences, University of Buenos Aires, Buenos Aires, Argentina.
  • Galigniana MD; Department of Biological Chemistry, Faculty of Natural Sciences, University of Buenos Aires, Buenos Aires, Argentina; Institute of Experimental Biology and Medicine-CONICET, Buenos Aires, Argentina.
  • Subrahmanyam CV; Department of Pharmaceutical Chemistry, Gokaraju Rangaraju College of Pharmacy, Osmania University, Hyderabad, India.
  • Gowrishankar NL; Swami Vivekananda Institute of Pharmaceutical Sciences, Nalgonda, Andhra Pradesh, India.
  • Raghavendra NM; Department of Pharmaceutical Chemistry, Gokaraju Rangaraju College of Pharmacy, Osmania University, Hyderabad, India.
Int J Biol Macromol ; 80: 253-9, 2015 09.
Article em En | MEDLINE | ID: mdl-26116388

Texto completo: 1 Base de dados: MEDLINE Assunto principal: Desenho de Fármacos / Proteínas de Choque Térmico HSP90 / Simulação de Acoplamento Molecular / Antineoplásicos Tipo de estudo: Prognostic_studies Limite: Humans Idioma: En Ano de publicação: 2015 Tipo de documento: Article

Texto completo: 1 Base de dados: MEDLINE Assunto principal: Desenho de Fármacos / Proteínas de Choque Térmico HSP90 / Simulação de Acoplamento Molecular / Antineoplásicos Tipo de estudo: Prognostic_studies Limite: Humans Idioma: En Ano de publicação: 2015 Tipo de documento: Article