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Fragment-Based Drug Discovery Targeting Inhibitor of Apoptosis Proteins: Discovery of a Non-Alanine Lead Series with Dual Activity Against cIAP1 and XIAP.
Chessari, Gianni; Buck, Ildiko M; Day, James E H; Day, Philip J; Iqbal, Aman; Johnson, Christopher N; Lewis, Edward J; Martins, Vanessa; Miller, Darcey; Reader, Michael; Rees, David C; Rich, Sharna J; Tamanini, Emiliano; Vitorino, Marc; Ward, George A; Williams, Pamela A; Williams, Glyn; Wilsher, Nicola E; Woolford, Alison J-A.
Afiliação
  • Chessari G; Astex Pharmaceuticals , 436 Cambridge Science Park, Milton Road, Cambridge, CB4 0QA, United Kingdom.
  • Buck IM; Astex Pharmaceuticals , 436 Cambridge Science Park, Milton Road, Cambridge, CB4 0QA, United Kingdom.
  • Day JE; Astex Pharmaceuticals , 436 Cambridge Science Park, Milton Road, Cambridge, CB4 0QA, United Kingdom.
  • Day PJ; Astex Pharmaceuticals , 436 Cambridge Science Park, Milton Road, Cambridge, CB4 0QA, United Kingdom.
  • Iqbal A; Astex Pharmaceuticals , 436 Cambridge Science Park, Milton Road, Cambridge, CB4 0QA, United Kingdom.
  • Johnson CN; Astex Pharmaceuticals , 436 Cambridge Science Park, Milton Road, Cambridge, CB4 0QA, United Kingdom.
  • Lewis EJ; Astex Pharmaceuticals , 436 Cambridge Science Park, Milton Road, Cambridge, CB4 0QA, United Kingdom.
  • Martins V; Astex Pharmaceuticals , 436 Cambridge Science Park, Milton Road, Cambridge, CB4 0QA, United Kingdom.
  • Miller D; Astex Pharmaceuticals , 436 Cambridge Science Park, Milton Road, Cambridge, CB4 0QA, United Kingdom.
  • Reader M; Astex Pharmaceuticals , 436 Cambridge Science Park, Milton Road, Cambridge, CB4 0QA, United Kingdom.
  • Rees DC; Astex Pharmaceuticals , 436 Cambridge Science Park, Milton Road, Cambridge, CB4 0QA, United Kingdom.
  • Rich SJ; Astex Pharmaceuticals , 436 Cambridge Science Park, Milton Road, Cambridge, CB4 0QA, United Kingdom.
  • Tamanini E; Astex Pharmaceuticals , 436 Cambridge Science Park, Milton Road, Cambridge, CB4 0QA, United Kingdom.
  • Vitorino M; Astex Pharmaceuticals , 436 Cambridge Science Park, Milton Road, Cambridge, CB4 0QA, United Kingdom.
  • Ward GA; Astex Pharmaceuticals , 436 Cambridge Science Park, Milton Road, Cambridge, CB4 0QA, United Kingdom.
  • Williams PA; Astex Pharmaceuticals , 436 Cambridge Science Park, Milton Road, Cambridge, CB4 0QA, United Kingdom.
  • Williams G; Astex Pharmaceuticals , 436 Cambridge Science Park, Milton Road, Cambridge, CB4 0QA, United Kingdom.
  • Wilsher NE; Astex Pharmaceuticals , 436 Cambridge Science Park, Milton Road, Cambridge, CB4 0QA, United Kingdom.
  • Woolford AJ; Astex Pharmaceuticals , 436 Cambridge Science Park, Milton Road, Cambridge, CB4 0QA, United Kingdom.
J Med Chem ; 58(16): 6574-88, 2015 Aug 27.
Article em En | MEDLINE | ID: mdl-26218264

Texto completo: 1 Base de dados: MEDLINE Assunto principal: Fragmentos de Peptídeos / Proteínas Inibidoras de Apoptose / Proteínas Inibidoras de Apoptose Ligadas ao Cromossomo X / Antineoplásicos Limite: Animals / Humans Idioma: En Ano de publicação: 2015 Tipo de documento: Article

Texto completo: 1 Base de dados: MEDLINE Assunto principal: Fragmentos de Peptídeos / Proteínas Inibidoras de Apoptose / Proteínas Inibidoras de Apoptose Ligadas ao Cromossomo X / Antineoplásicos Limite: Animals / Humans Idioma: En Ano de publicação: 2015 Tipo de documento: Article