Optimization and Evaluation of 5-Styryl-Oxathiazol-2-one Mycobacterium tuberculosis Proteasome Inhibitors as Potential Antitubercular Agents.

Russo, Francesco; Gising, Johan; Åkerbladh, Linda; Roos, Annette K; Naworyta, Agata; Mowbray, Sherry L; Sokolowski, Anders; Henderson, Ian; Alling, Torey; Bailey, Mai A; Files, Megan; Parish, Tanya; Karlén, Anders; Larhed, Mats

Russo, Francesco; Gising, Johan; Åkerbladh, Linda; Roos, Annette K; Naworyta, Agata; Mowbray, Sherry L; Sokolowski, Anders; Henderson, Ian; Alling, Torey; Bailey, Mai A; Files, Megan; Parish, Tanya; Karlén, Anders; Larhed, Mats.

Afiliação

Russo F; Department of Medicinal Chemistry, Organic Pharmaceutical Chemistry, BMC, Uppsala University Box 574, 751 23, Uppsala, Sweden.
Gising J; Department of Medicinal Chemistry, Organic Pharmaceutical Chemistry, BMC, Uppsala University Box 574, 751 23, Uppsala, Sweden.
Åkerbladh L; Department of Medicinal Chemistry, Organic Pharmaceutical Chemistry, BMC, Uppsala University Box 574, 751 23, Uppsala, Sweden.
Roos AK; Department of Cell and Molecular Biology, Science for Life Laboratory, BMC, Uppsala University Box 596, 751 24, Uppsala, Sweden.
Naworyta A; Department of Cell and Molecular Biology, BMC, Uppsala University Box 596, 751 24, Uppsala, Sweden.
Mowbray SL; Department of Cell and Molecular Biology, Science for Life Laboratory, BMC, Uppsala University Box 596, 751 24, Uppsala, Sweden.
Sokolowski A; Department of Medicinal Chemistry, Organic Pharmaceutical Chemistry, BMC, Uppsala University Box 574, 751 23, Uppsala, Sweden.
Henderson I; Medivir AB PO Box 1086, 141 22, Huddinge, Sweden.
Alling T; TB Discovery Research, Infectious Disease Research Institute Seattle, WA, 98102, USA.
Bailey MA; TB Discovery Research, Infectious Disease Research Institute Seattle, WA, 98102, USA.
Files M; TB Discovery Research, Infectious Disease Research Institute Seattle, WA, 98102, USA.
Parish T; TB Discovery Research, Infectious Disease Research Institute Seattle, WA, 98102, USA.
Karlén A; Department of Medicinal Chemistry, Organic Pharmaceutical Chemistry, BMC, Uppsala University Box 574, 751 23, Uppsala, Sweden.
Larhed M; Department of Medicinal Chemistry, Science for Life Laboratory, BMC, Uppsala University Box 574, 751 23, Uppsala, Sweden.