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Structure-Activity Study of Bioisosteric Trifluoromethyl and Pentafluorosulfanyl Indole Inhibitors of the AAA ATPase p97.
Alverez, Celeste; Arkin, Michelle R; Bulfer, Stacie L; Colombo, Raffaele; Kovaliov, Marina; LaPorte, Matthew G; Lim, Chaemin; Liang, Mary; Moore, William J; Neitz, R Jeffrey; Yan, Yongzhao; Yue, Zhizhou; Huryn, Donna M; Wipf, Peter.
Afiliação
  • Alverez C; Department of Pharmaceutical Sciences, University of Pittsburgh , Pittsburgh, Pennsylvania 15261, United States ; Chemical Diversity Center, University of Pittsburgh , Pittsburgh, Pennsylvania 15260, United States.
  • Arkin MR; Department of Pharmaceutical Chemistry, Small Molecule Discovery Center, University of California , San Francisco, California 94158, United States.
  • Bulfer SL; Department of Pharmaceutical Chemistry, Small Molecule Discovery Center, University of California , San Francisco, California 94158, United States.
  • Colombo R; Chemical Diversity Center, University of Pittsburgh , Pittsburgh, Pennsylvania 15260, United States.
  • Kovaliov M; Chemical Diversity Center, University of Pittsburgh , Pittsburgh, Pennsylvania 15260, United States.
  • LaPorte MG; Chemical Diversity Center, University of Pittsburgh , Pittsburgh, Pennsylvania 15260, United States.
  • Lim C; Chemical Diversity Center, University of Pittsburgh , Pittsburgh, Pennsylvania 15260, United States.
  • Liang M; Chemical Diversity Center, University of Pittsburgh , Pittsburgh, Pennsylvania 15260, United States.
  • Moore WJ; Leidos Biomedical Research, Inc. , Frederick, Maryland 21702, United States.
  • Neitz RJ; Department of Pharmaceutical Chemistry, Small Molecule Discovery Center, University of California , San Francisco, California 94158, United States.
  • Yan Y; Chemical Diversity Center, University of Pittsburgh , Pittsburgh, Pennsylvania 15260, United States.
  • Yue Z; Chemical Diversity Center, University of Pittsburgh , Pittsburgh, Pennsylvania 15260, United States.
  • Huryn DM; Department of Pharmaceutical Sciences, University of Pittsburgh , Pittsburgh, Pennsylvania 15261, United States ; Chemical Diversity Center, University of Pittsburgh , Pittsburgh, Pennsylvania 15260, United States.
  • Wipf P; Department of Pharmaceutical Sciences, University of Pittsburgh , Pittsburgh, Pennsylvania 15261, United States ; Chemical Diversity Center, University of Pittsburgh , Pittsburgh, Pennsylvania 15260, United States.
ACS Med Chem Lett ; 6(12): 1225-30, 2015 Dec 10.
Article em En | MEDLINE | ID: mdl-26713109

Texto completo: 1 Base de dados: MEDLINE Idioma: En Ano de publicação: 2015 Tipo de documento: Article

Texto completo: 1 Base de dados: MEDLINE Idioma: En Ano de publicação: 2015 Tipo de documento: Article