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Design and development of histone deacetylase (HDAC) chemical probes for cell-based profiling.
Albrow, Victoria E; Grimley, Rachel L; Clulow, James; Rose, Colin R; Sun, Jianmin; Warmus, Joseph S; Tate, Edward W; Jones, Lyn H; Storer, R Ian.
Afiliação
  • Albrow VE; Pfizer Ltd, The Portway Building, Granta Park, Great Abington, Cambridge, CB21 6GS, UK.
  • Grimley RL; Pfizer Ltd, The Portway Building, Granta Park, Great Abington, Cambridge, CB21 6GS, UK.
  • Clulow J; Department of Chemistry and Institute of Chemical Biology, Imperial College London, London, SW7 2AZ, UK.
  • Rose CR; Worldwide Medicinal Chemistry, Pfizer Inc., Eastern Point Road, Groton, Connecticut 06340, USA.
  • Sun J; Worldwide Medicinal Chemistry, Pfizer Inc., Eastern Point Road, Groton, Connecticut 06340, USA.
  • Warmus JS; Worldwide Medicinal Chemistry, Pfizer Inc., Eastern Point Road, Groton, Connecticut 06340, USA.
  • Tate EW; Department of Chemistry and Institute of Chemical Biology, Imperial College London, London, SW7 2AZ, UK.
  • Jones LH; Worldwide Medicinal Chemistry, Pfizer Inc., 610 Main Street, Cambridge, MA 02139, USA.
  • Storer RI; Worldwide Medicinal Chemistry, Pfizer Ltd, The Portway Building, Granta Park, Great Abington, Cambridge, CB21 6GS, UK. ian.storer@pfizer.com.
Mol Biosyst ; 12(6): 1781-9, 2016 05 24.
Article em En | MEDLINE | ID: mdl-27021930

Texto completo: 1 Base de dados: MEDLINE Assunto principal: Sondas Moleculares / Proteômica / Inibidores de Histona Desacetilases / Histona Desacetilases Limite: Humans Idioma: En Ano de publicação: 2016 Tipo de documento: Article

Texto completo: 1 Base de dados: MEDLINE Assunto principal: Sondas Moleculares / Proteômica / Inibidores de Histona Desacetilases / Histona Desacetilases Limite: Humans Idioma: En Ano de publicação: 2016 Tipo de documento: Article