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Surface plasmon resonance biosensor assay for the analysis of small-molecule inhibitor binding to human and parasitic phosphodiesterases.
Siderius, Marco; Shanmugham, Anitha; England, Paul; van der Meer, Tiffany; Bebelman, Jan Paul; Blaazer, Antoni R; de Esch, Iwan J P; Leurs, Rob.
Afiliação
  • Siderius M; Amsterdam Institute of Molecules, Medicines and Systems (AIMMS), Division of Medicinal Chemistry, VU University Amsterdam, De Boelelaan 1083, 1081 HV Amsterdam, The Netherlands. Electronic address: m.siderius@vu.nl.
  • Shanmugham A; IOTA Pharmaceuticals, St. John's Innovation Centre, Cowley Road, Cambridge CB4 0WS, United Kingdom.
  • England P; IOTA Pharmaceuticals, St. John's Innovation Centre, Cowley Road, Cambridge CB4 0WS, United Kingdom.
  • van der Meer T; Amsterdam Institute of Molecules, Medicines and Systems (AIMMS), Division of Medicinal Chemistry, VU University Amsterdam, De Boelelaan 1083, 1081 HV Amsterdam, The Netherlands.
  • Bebelman JP; Amsterdam Institute of Molecules, Medicines and Systems (AIMMS), Division of Medicinal Chemistry, VU University Amsterdam, De Boelelaan 1083, 1081 HV Amsterdam, The Netherlands.
  • Blaazer AR; Amsterdam Institute of Molecules, Medicines and Systems (AIMMS), Division of Medicinal Chemistry, VU University Amsterdam, De Boelelaan 1083, 1081 HV Amsterdam, The Netherlands.
  • de Esch IJ; Amsterdam Institute of Molecules, Medicines and Systems (AIMMS), Division of Medicinal Chemistry, VU University Amsterdam, De Boelelaan 1083, 1081 HV Amsterdam, The Netherlands; IOTA Pharmaceuticals, St. John's Innovation Centre, Cowley Road, Cambridge CB4 0WS, United Kingdom.
  • Leurs R; Amsterdam Institute of Molecules, Medicines and Systems (AIMMS), Division of Medicinal Chemistry, VU University Amsterdam, De Boelelaan 1083, 1081 HV Amsterdam, The Netherlands; IOTA Pharmaceuticals, St. John's Innovation Centre, Cowley Road, Cambridge CB4 0WS, United Kingdom.
Anal Biochem ; 503: 41-9, 2016 06 15.
Article em En | MEDLINE | ID: mdl-27033007

Texto completo: 1 Base de dados: MEDLINE Assunto principal: Inibidores de Fosfodiesterase / Proteínas de Protozoários / 3',5'-AMP Cíclico Fosfodiesterases / Ressonância de Plasmônio de Superfície / Nucleotídeo Cíclico Fosfodiesterase do Tipo 4 / Bibliotecas de Moléculas Pequenas Tipo de estudo: Guideline Limite: Humans Idioma: En Ano de publicação: 2016 Tipo de documento: Article

Texto completo: 1 Base de dados: MEDLINE Assunto principal: Inibidores de Fosfodiesterase / Proteínas de Protozoários / 3',5'-AMP Cíclico Fosfodiesterases / Ressonância de Plasmônio de Superfície / Nucleotídeo Cíclico Fosfodiesterase do Tipo 4 / Bibliotecas de Moléculas Pequenas Tipo de estudo: Guideline Limite: Humans Idioma: En Ano de publicação: 2016 Tipo de documento: Article