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7-Substituted 2-Nitro-5,6-dihydroimidazo[2,1-b][1,3]oxazines: Novel Antitubercular Agents Lead to a New Preclinical Candidate for Visceral Leishmaniasis.
Thompson, Andrew M; O'Connor, Patrick D; Marshall, Andrew J; Yardley, Vanessa; Maes, Louis; Gupta, Suman; Launay, Delphine; Braillard, Stephanie; Chatelain, Eric; Franzblau, Scott G; Wan, Baojie; Wang, Yuehong; Ma, Zhenkun; Cooper, Christopher B; Denny, William A.
Afiliação
  • Thompson AM; Auckland Cancer Society Research Centre, School of Medical Sciences, The University of Auckland , Private Bag 92019, Auckland 1142, New Zealand.
  • O'Connor PD; Auckland Cancer Society Research Centre, School of Medical Sciences, The University of Auckland , Private Bag 92019, Auckland 1142, New Zealand.
  • Marshall AJ; Auckland Cancer Society Research Centre, School of Medical Sciences, The University of Auckland , Private Bag 92019, Auckland 1142, New Zealand.
  • Yardley V; Faculty of Infectious & Tropical Diseases, London School of Hygiene & Tropical Medicine , Keppel Street, London WC1E 7HT, United Kingdom.
  • Maes L; Laboratory for Microbiology, Parasitology and Hygiene, Faculty of Pharmaceutical, Biomedical and Veterinary Sciences, University of Antwerp , Universiteitsplein 1, B-2610 Antwerp, Belgium.
  • Gupta S; Division of Parasitology, CSIR-Central Drug Research Institute , Lucknow 226031, India.
  • Launay D; Drugs for Neglected Diseases initiative, 15 Chemin Louis Dunant, 1202 Geneva, Switzerland.
  • Braillard S; Drugs for Neglected Diseases initiative, 15 Chemin Louis Dunant, 1202 Geneva, Switzerland.
  • Chatelain E; Drugs for Neglected Diseases initiative, 15 Chemin Louis Dunant, 1202 Geneva, Switzerland.
  • Franzblau SG; Institute for Tuberculosis Research, College of Pharmacy, University of Illinois at Chicago , 833 South Wood Street, Chicago, Illinois 60612, United States.
  • Wan B; Institute for Tuberculosis Research, College of Pharmacy, University of Illinois at Chicago , 833 South Wood Street, Chicago, Illinois 60612, United States.
  • Wang Y; Institute for Tuberculosis Research, College of Pharmacy, University of Illinois at Chicago , 833 South Wood Street, Chicago, Illinois 60612, United States.
  • Ma Z; Global Alliance for TB Drug Development , 40 Wall Street, New York 10005, United States.
  • Cooper CB; Global Alliance for TB Drug Development , 40 Wall Street, New York 10005, United States.
  • Denny WA; Auckland Cancer Society Research Centre, School of Medical Sciences, The University of Auckland , Private Bag 92019, Auckland 1142, New Zealand.
J Med Chem ; 60(10): 4212-4233, 2017 05 25.
Article em En | MEDLINE | ID: mdl-28459575

Texto completo: 1 Base de dados: MEDLINE Assunto principal: Leishmania donovani / Leishmania infantum / Leishmaniose Visceral / Nitroimidazóis / Antiprotozoários Limite: Animals / Female / Humans / Male Idioma: En Ano de publicação: 2017 Tipo de documento: Article

Texto completo: 1 Base de dados: MEDLINE Assunto principal: Leishmania donovani / Leishmania infantum / Leishmaniose Visceral / Nitroimidazóis / Antiprotozoários Limite: Animals / Female / Humans / Male Idioma: En Ano de publicação: 2017 Tipo de documento: Article